SCHEMBL15577702

SCHEMBL15577702

NC(=O)[C@H](Cc1ccccc1)Nc1ccc2ccccc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FCER2 P06734 4/20 0.53
ELANE P08246 1/20 0.49
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PPARG P37231 2/20 0.47
PPARA Q07869 2/20 0.47
EPHX1 P07099 1/20 0.46
PPARD Q03181 1/20 0.46
MRGPRX4 Q96LA9 1/20 0.46
MAPT P10636 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CAPN1 P07384 1/20 0.45
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
MC5R P33032 2/20 0.45
MC1R Q01726 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2779293 0.88 PPARG (0.53) KDM4ELMNAGAAHTTSMN1; SMN2
SCHEMBL2779289 0.88 PPARG (0.53) KDM4ELMNAGAAHTTSMN1; SMN2
SCHEMBL30436738 0.83 ATM (0.51) LMNAGAAPPARGPPARAPPARD
SCHEMBL2722699 0.83 ELANE (0.53) FCER2ELANEPPARGEPHX1CYP1A2
SCHEMBL1053745 0.83 ELANE (0.53) FCER2ELANEPPARGEPHX1CYP1A2
SCHEMBL28085739 0.82 MAPT (0.52) FCER2ELANEKDM4EGAAEPHX1
SCHEMBL16599266 0.80 SYK (0.49) ELANEKDM4EGAAHTTSMN1; SMN2
SCHEMBL28085748 0.79 MAPK1 (0.49) FCER2ELANEGAASMN1; SMN2PPARG
SCHEMBL4522563 0.79 FPR2 (0.58) FCER2ELANESMN1; SMN2PPARGEPHX1
SCHEMBL27723701 0.79 FPR2 (0.58) FCER2ELANESMN1; SMN2PPARGEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2895482-A1 HIV PROTEASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2015-07-22 EP claimed
WO-2014043019-A1 HIV PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2014-03-20 WO claimed