SCHEMBL1558049

SCHEMBL1558049

COc1ccc(-c2ccccc2CCc2ccc3ccccc3n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54
NPC1 O15118 1/20 0.54
NFKB1 P19838 1/20 0.54
RAB9A P51151 1/20 0.54
NFKB2 Q00653 1/20 0.54
RELA Q04206 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
PDE10A Q9Y233 9/20 0.52
ACACA Q13085 1/20 0.43
LMNA P02545 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2E1 P05181 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C8 P10632 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28002003 0.80 MEN1 (0.55) KDM4EALDH1A1NPC1NFKB1RAB9A
SCHEMBL1424251 0.79 CYSLTR1 (0.58) PDE10ACYSLTR1CYSLTR2
SCHEMBL28002107 0.77 DHFR (0.58) SMN1; SMN2PDE10ACYP1A2
SCHEMBL1423762 0.75 CYSLTR1 (0.61) PDE10ACYSLTR1CYSLTR2
SCHEMBL13772898 0.75 CYSLTR1 (0.69) KDM4EALDH1A1NPC1NFKB1RAB9A
SCHEMBL17761067 0.74 NPC1 (0.59) KDM4EALDH1A1NPC1NFKB1RAB9A
SCHEMBL4375331 0.74 PPARA (0.53) NPC1RAB9ASMN1; SMN2LMNAL3MBTL1
SCHEMBL14911661 0.73 PDE10A (0.48) KDM4EALDH1A1NPC1NFKB1RAB9A
SCHEMBL14351769 0.73 PDE10A (0.48) KDM4EALDH1A1NPC1NFKB1RAB9A
SCHEMBL10547475 0.73 CYSLTR1 (0.76) PDE10ACYSLTR1CYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2303863-A1 5- AND 6-MEMBERED HETEROCYCLIC COMPOUNDS Envivo Pharmaceuticals, Inc. (US) 2011-04-06 EP disclosed