SCHEMBL28002003

SCHEMBL28002003

COc1ccc(CCc2ccc3ccccc3n2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54
NPC1 O15118 1/20 0.54
NFKB1 P19838 1/20 0.54
RAB9A P51151 1/20 0.54
NFKB2 Q00653 1/20 0.54
RELA Q04206 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
DHFR P00374 1/20 0.53
CYSLTR1 Q9Y271 5/20 0.51
FFAR1 O14842 1/20 0.51
AKR1B1 P15121 1/20 0.51
CYSLTR2 Q9NS75 4/20 0.50
PDE10A Q9Y233 4/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2E1 P05181 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C8 P10632 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30842277 0.86 NPC1 (0.55) MEN1KMT2AKDM4EALDH1A1NPC1
SCHEMBL18546229 0.84 FFAR1 (0.48) CYSLTR1FFAR1AKR1B1CYSLTR2PDE10A
SCHEMBL1557935 0.82 PTGS1 (0.53) MEN1KMT2AKDM4EALDH1A1NPC1
SCHEMBL3950944 0.81 KCNH2 (0.61) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL8588707 0.81 PKM (0.59) MEN1KMT2AKDM4EALDH1A1NPC1
SCHEMBL1558049 0.80 KDM4E (0.54) KDM4EALDH1A1NPC1NFKB1RAB9A
SCHEMBL10547475 0.79 CYSLTR1 (0.76) CYSLTR1FFAR1AKR1B1CYSLTR2PDE10A
SCHEMBL2913941 0.79 PDE10A (0.61) CYSLTR1CYSLTR2PDE10ACYP1A2CYP3A4
SCHEMBL15549053 0.79 CYSLTR1 (0.51) MEN1KMT2AKDM4EALDH1A1NPC1
SCHEMBL3270954 0.79 CYSLTR1 (0.56) MEN1KMT2ANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104529889-B A kind of dehydration C- alkylations of heterocyclic methyl compound 温州大学 2018-09-04 CN disclosed
CN-104529889-A Dehydration C-alkylation method for heterocyclic methyl compound UNIV WENZHOU 2015-04-22 CN disclosed