SCHEMBL15580702

SCHEMBL15580702

C=C(O)c1cnc(Oc2ccc([C@@H](C)[C@@](O)(c3ccc4c(c3)N(C)C(=O)CO4)C(F)(F)F)c(Cl)c2)cn1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 1/20 0.33
RIPK1 Q13546 2/20 0.32
SLC5A1 P13866 2/20 0.32
SLC5A2 P31639 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474528 0.94 GPR55 (0.33) GPR55RIPK1
SCHEMBL12164282 0.94 GPR55 (0.33) GPR55RIPK1
SCHEMBL474356 0.91 GPR55 (0.34) GPR55RIPK1
SCHEMBL12164280 0.91 GPR55 (0.34) GPR55RIPK1
SCHEMBL15520243 0.90 GPR55 (0.33) GPR55
SCHEMBL12164254 0.86 GPR55 (0.33) GPR55
SCHEMBL474020 0.86 HRH3 (0.38) GPR55
SCHEMBL12164240 0.86 HRH3 (0.38) GPR55
SCHEMBL474532 0.86 GPR55 (0.33) GPR55
SCHEMBL12163916 0.84 CMA1 (0.33) GPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP disclosed