SCHEMBL15599236

SCHEMBL15599236

CC(C)(C)OC(=O)c1cc(Cl)c(Oc2cnc(OCC(F)(F)F)c(Cl)c2)cc1F

nearest known ligand 0.60

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 0.60
SCN5A Q14524 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16175358 0.94 SCN9A (0.54) SCN9ASCN5A
SCHEMBL15544113 0.91 SCN9A (0.51) SCN9ASCN5A
SCHEMBL1690160 0.91 SCN9A (0.69) SCN9ASCN5A
SCHEMBL17244933 0.90 SCN9A (0.58) SCN9ASCN5A
SCHEMBL15599208 0.89 SCN9A (0.64) SCN9ASCN5A
SCHEMBL15543933 0.88 SCN9A (0.65) SCN9ASCN5A
SCHEMBL15558876 0.87 SCN9A (0.72) SCN9ASCN5A
SCHEMBL15542946 0.86 SCN9A (0.65) SCN9ASCN5A
SCHEMBL19411921 0.85 SCN9A (0.57) SCN9ASCN5A
SCHEMBL16175064 0.85 SCN9A (0.57) SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180346416-A1 N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2018-12-06 US disclosed
US-10071957-B2 N-substituted benzamides and methods of use thereof GENENTECH, INC. (US) 2018-09-11 US disclosed
EP-2870138-B1 N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF GENENTECH INC (US) 2018-08-22 EP disclosed
US-20150322002-A1 N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2015-11-12 US disclosed
US-20150322002-A1 N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2015-11-12 US disclosed
WO-2014008458-A2 N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2014-01-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150322002-A1 N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF BRIX1, SNRPD2, RDX SCN9A 1104/4885SCN5A 724/4885
US-10071957-B2 N-substituted benzamides and methods of use thereof BRIX1, SNRPD2, RDX SCN9A 1104/4885SCN5A 724/4885
US-20180346416-A1 N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF BRIX1, RDX, P2RX3 SCN9A 501/4885SCN5A 327/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.