SCHEMBL15599330

SCHEMBL15599330

Cc1cnc(NC(=O)OC(C)(C)C)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.39
LCK P06239 1/20 0.38
CYP17A1 P05093 1/20 0.38
HDAC6 Q9UBN7 1/20 0.37
DHODH Q02127 2/20 0.37
ATR Q13535 1/20 0.36
ACVR1B P36896 1/20 0.36
TGFBR1 P36897 1/20 0.36
ACVRL1 P37023 1/20 0.36
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
MAPKAPK2 P49137 1/20 0.36
EGLN2 Q96KS0 2/20 0.35
RORC P51449 2/20 0.35
MAPK1 P28482 1/20 0.35
S1PR3 Q99500 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5456915 0.87 SYK (0.46) SYKIRAK4CYP17A1ATRACVR1B
SCHEMBL7416577 0.85 LCK (0.45) LCKATRGSK3BDYRK1AMAPKAPK2
SCHEMBL30850163 0.84 ATR (0.39) SYKLCKCYP17A1ATRGSK3B
SCHEMBL2960307 0.84 AAK1 (0.43) SYKLCKCYP17A1HDAC6ATR
SCHEMBL17282546 0.84 SYK (0.42) SYKCYP17A1HDAC6ATRACVR1B
SCHEMBL23167942 0.83 HDAC6 (0.56) SYKHDAC6
SCHEMBL25138307 0.82 ATR (0.42) SYKLCKCYP17A1HDAC6ATR
SCHEMBL7412985 0.79 SYK (0.42) SYKLCKCYP17A1ATRGSK3B
SCHEMBL17017349 0.78 HCRTR1 (0.43) SYKHDAC6
SCHEMBL28490153 0.76 SYK (0.40) SYKCYP17A1ATRACVR1BTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014006554-A1 3-(PYRAZOLYL)-1H-PYRROLO[2,3-b]PYRIDINE DERIVATIVES AS KINASE INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2014-01-09 WO disclosed