SCHEMBL15616865

SCHEMBL15616865

Nc1cc2c(c(C(=O)I)c1)OCC2

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.51
HTR3A P46098 1/20 0.36
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
XDH P47989 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
CYP2A6 P11509 1/20 0.32
MAP2K1 Q02750 3/20 0.32
PI4K2A Q9BTU6 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
PTGES O14684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL727922 0.85 PARP1 (0.53) PARP1HTR3AMAPTNPSR1RXFP1
SCHEMBL30573216 0.85 PARP1 (0.53) PARP1HTR3AMAPTNPSR1RXFP1
SCHEMBL13294905 0.83 PARP1 (0.51) PARP1HTR3AMAPTNPSR1RXFP1
SCHEMBL8550081 0.74 PARP1 (0.43) PARP1MAPT
SCHEMBL8549330 0.74 L3MBTL4 (0.45) PARP1HTR3APTGS1PTGS2
SCHEMBL15427984 0.73 CYP3A4 (0.39) PARP1MAPTMAP2K1
SCHEMBL14686084 0.71 PARP1 (0.42) PARP1MAPTXDHSLC22A12CYP2A6
SCHEMBL9050184 0.70 PARP1 (0.39) PARP1
SCHEMBL1976575 0.69 PARP1 (0.46) PARP1
SCHEMBL7484709 0.69 PARP1 (0.39) PARP1CYP2A6PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014041140-A1 METHODS OF TREATING HAIR RELATED CONDITIONS NOGRA PHARMA LIMITED (IE) 2014-03-20 WO disclosed