SCHEMBL8549330

SCHEMBL8549330

CN(C)CCC(=O)c1cc(N)cc2c1OCC2

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
L3MBTL4 Q8NA19 1/20 0.45
PARP1 P09874 2/20 0.43
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
MAOB P27338 3/20 0.36
MAOA P21397 1/20 0.36
CHEK1 O14757 1/20 0.34
CHEK2 O96017 1/20 0.34
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
STAT6 P42226 1/20 0.33
HSD17B10 Q99714 1/20 0.33
THRB P10828 4/20 0.32
THRA P10827 3/20 0.32
HTR3A P46098 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13294905 0.77 PARP1 (0.51) PARP1PTGS1PTGS2ALDH1A1HSD17B10
SCHEMBL9050184 0.75 PARP1 (0.39) PARP1
SCHEMBL727922 0.75 PARP1 (0.53) PARP1PTGS2ALDH1A1CYP3A4CYP2C9
SCHEMBL30573216 0.75 PARP1 (0.53) PARP1PTGS2ALDH1A1CYP3A4CYP2C9
SCHEMBL15616865 0.74 PARP1 (0.51) PARP1PTGS1PTGS2HTR3A
SCHEMBL8550081 0.74 PARP1 (0.43) PARP1ALDH1A1CYP1A2
SCHEMBL8551730 0.72 NOS1 (0.34) PARP1PTGS1PTGS2
SCHEMBL8550551 0.70 HTR1B (0.41)
SCHEMBL8551468 0.67 KCNH2 (0.35) PARP1
SCHEMBL8551471 0.67 KCNH2 (0.35) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736025-B1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT1D ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1998-07-22 EP disclosed
US-5700818-A Dihydrobenzofuranyl-biphenyl carboxamides having 5HT1D antagonistic activity SMITHKLINE BEECHAM P.L.C. (GB) 1997-12-23 US disclosed
EP-0736025-A1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT 1D? ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1996-10-09 EP disclosed
WO-1995017401-A1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT1D ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1995-06-29 WO disclosed