SCHEMBL156346

SCHEMBL156346

O=C(O)c1ccc(Br)cc1F

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.68
KDM4E B2RXH2 1/20 0.53
GLA P06280 1/20 0.53
NPC1 O15118 2/20 0.51
ALDH1A1 P00352 2/20 0.51
LMNA P02545 2/20 0.51
RAB9A P51151 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
KMT2A Q03164 2/20 0.51
GAA P10253 1/20 0.51
FLT1 P17948 1/20 0.46
FLT4 P35916 1/20 0.46
KDR P35968 1/20 0.46
TMEM97 Q5BJF2 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
MAP2K1 Q02750 1/20 0.44
MYC P01106 1/20 0.44
NR4A1 P22736 1/20 0.44
GPR27 Q9NS67 1/20 0.44
CES2 O00748 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2349044 0.98 DGAT1 (0.66) DGAT1KDM4EGLANPC1ALDH1A1
Bromide SCHEMBL25212853 0.86 DGAT1 (0.53) DGAT1KDM4EGLANPC1ALDH1A1
SCHEMBL6222444 0.86 RARB (0.56) DGAT1KDM4EGLALMNARXFP1
SCHEMBL4464312 0.84 DGAT1 (0.70) DGAT1KDM4EGLANPC1ALDH1A1
SCHEMBL25379561 0.83 DGAT1 (0.50) DGAT1KDM4EGLANPC1ALDH1A1
SCHEMBL6818016 0.83 DGAT1 (0.63) DGAT1KDM4EGLANPC1ALDH1A1
SCHEMBL2554 0.83 KDM4E (0.59) DGAT1KDM4EGLANPC1ALDH1A1
SCHEMBL30722862 0.83 KDM4E (0.59) DGAT1KDM4EGLANPC1ALDH1A1
SCHEMBL2095201 0.81 DGAT1 (0.66) DGAT1KDM4EGLANPC1ALDH1A1
SCHEMBL321094 0.81 DGAT1 (0.66) DGAT1KDM4EGLANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2173 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118955313-B Synthesis method of enzalutamide key intermediate 安徽峆一药业股份有限公司 2025-06-17 CN claimed
CN-117820218-B Preparation method of apatamide and intermediate 江苏希迪制药有限公司 2025-05-27 CN claimed
CN-118955313-A Synthesis method of enzalutamide key intermediate 安徽峆一药业股份有限公司 2024-11-15 CN claimed
CN-117820306-A Axial chiral luminescent material with double luminescent centers and preparation method and application thereof 南通大学 2024-04-05 CN claimed
CN-117820218-A Preparation method of apatamide and intermediate 江苏希迪制药有限公司 2024-04-05 CN claimed
CN-117534652-A Preparation method of apatamide 黄冈人福药业有限责任公司 2024-02-09 CN claimed
CN-116903646-A Axial chiral boron-nitrogen luminescent material and preparation method and application thereof 南通大学 2023-10-20 CN claimed
CN-115215791-B Solvent-free preparation method of organic eutectic material 北京仿生界面科学未来技术研究院 2023-10-03 CN claimed
US-20230159524-A1 METHODS FOR SYNTHESIZING N-(PHENYLSULFONYL)BENZAMIDE COMPOUNDS AND INTERMEDIATES THEREOF ASCENTAGE PHARMA (SUZHOU) CO., LTD. (CN) 2023-05-25 US claimed
CN-113698310-B Preparation method of enzalutamide diester intermediate 江西金丰药业有限公司 2023-03-17 CN claimed
CN-105753802-B 3- isopropyl -6- bromine benzoisoxazoles and preparation method thereof 广东环境保护工程职业学院 2018-06-05 CN claimed
US-20170190670-A1 IMPROVED PROCESS FOR THE PREPARATION OF ENZALUTAMIDE SHILPA MEDICARE LIMITED (IN) 2017-07-06 US claimed
EP-3168214-A1 SUBSTITUTED 2-THIOXO-IMIDAZOLIDIN-4-ONES AND SPIRO ANALOGUES THEREOF, ACTIVE ANTI-CANCER INGREDIENT, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION, METHOD FOR TREATING PROSTATE CANCER R-PHHARM OVERSEAS INK. (US) 2017-05-17 EP claimed
EP-3166931-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF ENZALUTAMIDE Shilpa Medicare Limited (IN) 2017-05-17 EP claimed
CN-105936633-A 5-(3-isopropyl benzisoxazol)pyrazin-2-amine and preparation method thereof 广东环境保护工程职业学院 2016-09-14 CN claimed
CN-105753802-A 3-isopropyl-6-bromine benzisoxazole and preparing method thereof 广东环境保护工程职业学院 2016-07-13 CN claimed
WO-2016005875-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF ENZALUTAMIDE SHILPA MEDICARE LIMITED (IN) 2016-01-14 WO claimed
CN-101543943-B Leadless rosin core low-halogen no-clean scaling powder and method for preparing same YUNNAN TIN COMPANY GROUP HOLDING CO LTD 2012-07-11 CN claimed
CN-101543943-A Leadless rosin core low-halogen no-clean scaling powder and method for preparing same YUNNAN TIN COMPANY GROUP HOLDI 2009-09-30 CN claimed
EP-1377589-B1 OXAZOLYL-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS PHARMACIA ITALIA SPA (IT) 2005-09-07 EP claimed