SCHEMBL15664001

SCHEMBL15664001

Cc1ccc(Nc2cccnc2C)c(OC(=O)Nc2ccn(C)n2)n1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.40
PDE4D Q08499 2/20 0.39
NOTUM Q6P988 1/20 0.39
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
PIK3CA P42336 2/20 0.37
MTOR P42345 2/20 0.37
GRM5 P41594 2/20 0.37
PDE10A Q9Y233 1/20 0.37
GCK P35557 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
MAPT P10636 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
LPAR1 Q92633 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15663798 0.86 NPC1 (0.44) NOTUMNPC1RAB9APIK3CAMTOR
SCHEMBL15663956 0.85 PDE10A (0.38) NOTUMNPC1RAB9APIK3CAMTOR
SCHEMBL15663618 0.83 PDE10A (0.43) NOTUMNPC1RAB9APIK3CAMTOR
SCHEMBL15663440 0.83 GRM5 (0.49) NOTUMNPC1RAB9APIK3CAMTOR
SCHEMBL5201513 0.82 PDE10A (0.53) PDE4BPDE4DNOTUMNPC1RAB9A
SCHEMBL15663415 0.82 HPGDS (0.38) NOTUMNPC1RAB9AGRM5PDE10A
SCHEMBL15663961 0.82 PDE10A (0.39) NOTUMNPC1RAB9APIK3CAMTOR
SCHEMBL15664200 0.81 LPAR1 (0.34) NPC1RAB9AGRM5HTTMAPT
SCHEMBL15663513 0.81 NPC1 (0.38) NOTUMNPC1RAB9APIK3CAMTOR
SCHEMBL15663526 0.80 GRM5 (0.40) PDE4DGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1858854-B1 PYRIDINE-2-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2014-05-07 EP claimed