E626

E626

SCHEMBL15670533

NC(CC(=O)O)C(=O)O.Nc1nc2c(ncn2[C@@H]2O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]2O)c(=O)[nH]1

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC6A2SLC6A3

The experimentally established mechanism targets of E626. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.70
IMPDH2 P12268 7/20 0.67
TGM2 P21980 1/20 0.65
IMPDH1 P20839 2/20 0.64
TAS1R3 Q7RTX0 2/20 0.64
TAS1R1 Q7RTX1 2/20 0.64
KRAS P01116 8/20 0.61
HINT1 P49773 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
E626 SCHEMBL15670526 0.94 NT5E (0.69) NT5EIMPDH2TGM2IMPDH1TAS1R3
E626 SCHEMBL15670415 0.93 NT5E (0.71) NT5EIMPDH2TGM2IMPDH1TAS1R3
E626 SCHEMBL15670776 0.92 NT5E (0.60) NT5EIMPDH2TGM2IMPDH1TAS1R3
E626 SCHEMBL15670774 0.92 NT5E (0.70) NT5EIMPDH2TGM2IMPDH1TAS1R3
E626 SCHEMBL15670587 0.91 NT5E (0.69) NT5EIMPDH2TGM2IMPDH1TAS1R3
E626 SCHEMBL15670515 0.91 NT5E (0.75) NT5EIMPDH2TGM2IMPDH1TAS1R3
E626 SCHEMBL18759049 0.91 NT5E (0.83) NT5EIMPDH2TGM2IMPDH1TAS1R3
E626 SCHEMBL20677331 0.91 NT5E (0.83) NT5EIMPDH2TGM2IMPDH1TAS1R3
E626 SCHEMBL20276926 0.91 NT5E (0.83) NT5EIMPDH2TGM2IMPDH1TAS1R3
E626 SCHEMBL21163348 0.91 NT5E (0.83) NT5EIMPDH2TGM2IMPDH1TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2914132-A1 FLAVOUR ADDITIVES Mars, Incorporated (US) 2015-09-09 EP disclosed
WO-2014068045-A1 FLAVOUR ADDITIVES MARS, INCORPORATED (US) 2014-05-08 WO disclosed