SCHEMBL15701100

SCHEMBL15701100

COc1ccc(Cl)cc1C(C)C(=O)Nc1ccc2nc(NC(=O)c3cscn3)sc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.55
DCLK1 O15075 1/20 0.49
FES P07332 1/20 0.49
PIM1 P11309 1/20 0.49
CDK2 P24941 1/20 0.49
GSK3A P49840 1/20 0.49
GSK3B P49841 1/20 0.49
IRAK1 P51617 1/20 0.49
MAP4K2 Q12851 1/20 0.49
NTRK3 Q16288 1/20 0.49
HIPK4 Q8NE63 1/20 0.49
AURKB Q96GD4 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
STK17A Q9UEE5 1/20 0.49
MAP4K5 Q9Y4K4 1/20 0.49
CSNK1G3 Q9Y6M4 1/20 0.49
KDM4E B2RXH2 3/20 0.48
NPSR1 Q6W5P4 2/20 0.48
GAA P10253 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17148443 0.97 NTRK1 (0.53) NTRK1DCLK1FESPIM1CDK2
SCHEMBL15701126 0.89 NTRK1 (0.45) NTRK1DCLK1FESPIM1CDK2
SCHEMBL15701165 0.83 ACP1 (0.46) NTRK1KDM4ECASP3SENP7SENP8
SCHEMBL15701281 0.80 MAPT (0.64) NTRK1KDM4ENPSR1RXFP1NPC1
SCHEMBL15701028 0.80 RAB9A (0.48) NTRK1KDM4ECASP3SENP7SENP8
SCHEMBL15701026 0.80 RAB9A (0.48) NTRK1KDM4ECASP3SENP7SENP8
SCHEMBL15701139 0.78 DYRK1A (0.42) NTRK1KDM4ECASP3SENP7SENP8
SCHEMBL15701057 0.78 CASP3 (0.45) NTRK1KDM4ENPSR1CASP3SENP7
SCHEMBL19446717 0.78 RAB9A (0.52) KDM4ERXFP1CASP3SENP7SENP8
SCHEMBL15701278 0.77 CASP3 (0.50) KDM4ECASP3SENP7SENP8SENP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2914592-B1 INHIBITORS OF CYTOMEGALOVIRUS BOEHRINGER INGELHEIM INT (DE) 2017-10-11 EP disclosed
WO-2014070979-A1 INHIBITORS OF CYTOMEGALOVIRUS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-05-08 WO disclosed