SCHEMBL15733247

SCHEMBL15733247

Cc1nc(N2CCOCC2)cc(N(C)C)c1C(=O)NCc1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAPEPLD Q6IQ20 2/20 0.48
THRB P10828 2/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 3/20 0.45
RXFP1 Q9HBX9 1/20 0.44
TSHR P16473 2/20 0.44
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TP53 P04637 1/20 0.44
PIK3CB P42338 3/20 0.43
USP2 O75604 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
KLKB1 P03952 1/20 0.43
KLK1 P06870 1/20 0.43
POLB P06746 1/20 0.43
PIK3CA P42336 1/20 0.42
PIK3CD O00329 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15735460 0.85 THRB (0.48) NAPEPLDTHRBMEN1KMT2ALMNA
SCHEMBL2132334 0.85 MEN1 (0.52) NAPEPLDTHRBMEN1KMT2ALMNA
SCHEMBL15733276 0.84 NAPEPLD (0.47) NAPEPLDTHRBMEN1KMT2ALMNA
SCHEMBL15733146 0.84 THRB (0.49) NAPEPLDTHRBMEN1KMT2ALMNA
SCHEMBL15735333 0.83 THRB (0.47) NAPEPLDTHRBMEN1KMT2ALMNA
SCHEMBL15733200 0.83 KDM4E (0.48) NAPEPLDTHRBMEN1KMT2ALMNA
SCHEMBL2130234 0.80 MEN1 (0.49) NAPEPLDTHRBMEN1KMT2ALMNA
SCHEMBL2129573 0.79 MEN1 (0.52) NAPEPLDTHRBMEN1KMT2ALMNA
SCHEMBL2131731 0.79 MEN1 (0.52) NAPEPLDTHRBMEN1KMT2ALMNA
SCHEMBL2131202 0.79 MEN1 (0.52) NAPEPLDTHRBMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925316-A1 SUBSTITUTED AMINO-ARYLCARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2015-10-07 EP claimed
WO-2014082739-A1 SUBSTITUTED AMINO-ARYLCARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2014-06-05 WO claimed
US-20140148454-A1 SUBSTITUTED AMINO-ACRYLCARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2014-05-29 US claimed
EP-4584250-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS Biohaven Therapeutics Ltd. (VG) 2025-07-16 EP disclosed
EP-4580679-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS AND NMDA RECEPTOR ANTAGONISTS Biohaven Therapeutics Ltd. (VG) 2025-07-09 EP disclosed
WO-2024054807-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS AND TDP-43 MODULATORS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-14 WO disclosed
WO-2024054811-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-14 WO disclosed
WO-2024050389-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS AND NMDA RECEPTOR ANTAGONISTS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-07 WO disclosed
EP-2925316-A1 SUBSTITUTED AMINO-ARYLCARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2015-10-07 EP disclosed
WO-2014082739-A1 SUBSTITUTED AMINO-ARYLCARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2014-06-05 WO disclosed
US-20140148454-A1 SUBSTITUTED AMINO-ACRYLCARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2014-05-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140148454-A1 SUBSTITUTED AMINO-ACRYLCARBOXAMIDES AS KCNQ2/3 MODULATORS KCNJ2, KCNQ1, KCNQ2 NAPEPLD 869/4885THRB 1687/4885MEN1 4240/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.