SCHEMBL15739482

SCHEMBL15739482

CCN(CC1CCCC1)c1nc2ccccc2cc1CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C1=NN(C)NN1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.32
SGMS1 Q86VZ5 1/20 0.31
SGMS2 Q8NHU3 1/20 0.31
APAF1 O14727 2/20 0.30
UBE2N P61088 2/20 0.30
NPSR1 Q6W5P4 2/20 0.30
BCHE P06276 1/20 0.30
ACHE P22303 1/20 0.30
IDE P14735 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15739490 0.98 CRHR1 (0.31) TACR1
SCHEMBL15981331 0.97 CRHR1 (0.32)
SCHEMBL15739506 0.88 LMNA (0.33) TACR1
SCHEMBL14389954 0.88
SCHEMBL5624474 0.84 TACR1 (0.33) TACR1SGMS1SGMS2BCHEACHE
SCHEMBL5623860 0.83 TACR1 (0.33) TACR1SGMS1SGMS2APAF1UBE2N
SCHEMBL4361019 0.83 CETP (0.38)
SCHEMBL15981910 0.83 CETP (0.31) TACR1UBE2NIDE
SCHEMBL5626270 0.82 TACR1 (0.32) TACR1SGMS1SGMS2BCHEACHE
SCHEMBL15739594 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014128564-A2 PHARMACEUTICAL COMPOSITIONS OF CETP INHIBITORS DR. REDDY'S LABORATORIES LTD. (IN) 2014-08-28 WO disclosed
WO-2014076568-A2 PHARMACEUTICAL COMPOSITIONS OF CETP INHIBITORS DR. REDDY'S LABORATORIES LTD. (IN) 2014-05-22 WO disclosed