SCHEMBL15740475

SCHEMBL15740475

O=CC(OC1CCC(Nc2ccc([N+](=O)[O-])c(C(F)(F)F)c2)CC1)N1CCN(Cc2ccc3cc(C(F)(F)F)ccc3n2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MCHR1 Q99705 2/20 0.37
TMEM97 Q5BJF2 8/20 0.34
CXCR3 P49682 1/20 0.33
HTR2C P28335 1/20 0.31
SERPINE1 P05121 1/20 0.31
ROCK2 O75116 1/20 0.31
CES2 O00748 1/20 0.31
ABCB11 O95342 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
GLA P06280 1/20 0.31
CYP3A4 P08684 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
AR P10275 1/20 0.31
CHRM1 P11229 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15740437 0.95 MAPK1 (0.38) MAPK1NPSR1MCHR1TMEM97CXCR3
SCHEMBL15740426 0.88 HRH3 (0.42) MAPK1NPSR1MCHR1TMEM97SERPINE1
SCHEMBL15740442 0.88 MAPK1 (0.39) MAPK1NPSR1MCHR1TMEM97HTR2C
SCHEMBL15740454 0.88 TMEM97 (0.37) MAPK1NPSR1TMEM97SERPINE1ROCK2
SCHEMBL15740432 0.85 MAPK1 (0.36) MAPK1NPSR1TMEM97SERPINE1ROCK2
SCHEMBL15740430 0.85 MAPK1 (0.37) MAPK1NPSR1TMEM97SERPINE1CES2
SCHEMBL15740364 0.84 SIRT6 (0.41) MAPK1NPSR1TMEM97SERPINE1CES2
SCHEMBL15707912 0.84 MCHR1 (0.42) MAPK1NPSR1MCHR1TMEM97CXCR3
SCHEMBL15727599 0.84 MCHR1 (0.42) MAPK1NPSR1MCHR1TMEM97CXCR3
SCHEMBL15740443 0.83 TMEM97 (0.37) MAPK1NPSR1TMEM97CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922845-A2 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF Merial, Inc. (US) 2015-09-30 EP disclosed
WO-2014081697-A2 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF MERIAL LIMITED (US) 2014-05-30 WO disclosed