SCHEMBL1574475

SCHEMBL1574475

NC[C@@H](NC(=O)C1CN(C(=O)O)C1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 7/20 0.46
RPS6KA5 O75582 2/20 0.43
AKT1 P31749 2/20 0.43
GSK3B P49841 2/20 0.43
NEK4 P51957 2/20 0.43
PRKCD Q05655 2/20 0.43
PRKG2 Q13237 2/20 0.43
ROCK1 Q13464 2/20 0.43
PRKG1 Q13976 2/20 0.43
PKN2 Q16513 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
MAPK13 O15264 1/20 0.43
DYRK3 O43781 1/20 0.43
ROCK2 O75116 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
CHEK2 O96017 1/20 0.43
PRKCG P05129 1/20 0.43
CDK1 P06493 1/20 0.43
PIM1 P11309 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1574176 0.89 CCR5 (0.58) CCR5RPS6KA5AKT1GSK3BNEK4
SCHEMBL1574502 0.87 CCR5 (0.46) CCR5ITGB3ITGA2BF2RF11
SCHEMBL515734 0.81 RECQL (0.61) CCR5LMNAF11RECQL
SCHEMBL1573549 0.80 RPS6KA5 (0.45) RPS6KA5AKT1GSK3BNEK4PRKCD
SCHEMBL115980 0.73 ROCK1 (0.55) RPS6KA5AKT1GSK3BNEK4PRKCD
SCHEMBL4598191 0.73 ROCK1 (0.55) RPS6KA5AKT1GSK3BNEK4PRKCD
SCHEMBL4697349 0.73 CCR5 (0.84) CCR5
SCHEMBL1574310 0.72 CCR5 (0.44) CCR5RPS6KA5AKT1GSK3BNEK4
Hydrochloric Acid SCHEMBL7973435 0.72 RPS6KA5 (0.54) RPS6KA5AKT1GSK3BNEK4PRKCD
SCHEMBL8652164 0.72 RPS6KA5 (0.54) RPS6KA5AKT1GSK3BNEK4PRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140085-B1 AZABICYCLOALKANES AS CCR5 MODULATORS PHIVCO UK LTD (GB) 2011-04-13 EP disclosed