SCHEMBL1574748

SCHEMBL1574748

CN(C)C1CN(C(=O)Nc2cccc(C(F)(F)F)c2)C1

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 6/20 0.63
TP53 P04637 1/20 0.59
RAB9A P51151 3/20 0.56
POLB P06746 1/20 0.56
LMNA P02545 3/20 0.55
MAPT P10636 2/20 0.55
GAA P10253 1/20 0.55
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
HTT P42858 2/20 0.52
EPHX2 P34913 1/20 0.52
CCR2 P41597 1/20 0.51
KCNH2 Q12809 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1574917 0.87 GRIN2B (0.63) GRIN2BTP53RAB9APOLBLMNA
SCHEMBL1575005 0.87 GRIN2B (0.49) GRIN2BLMNAMAPT
SCHEMBL1574854 0.86 GRIN2B (0.59) GRIN2BTP53RAB9APOLBLMNA
SCHEMBL1574819 0.86 GRIN2B (0.59) GRIN2BTP53RAB9APOLBLMNA
SCHEMBL1574907 0.84 GRIN2B (0.57) GRIN2BTP53RAB9APOLBLMNA
SCHEMBL1575047 0.84 CYP2D6 (0.55) POLBMAPT
SCHEMBL14433872 0.84 GRIN2B (0.61) GRIN2BTP53RAB9ALMNAMAPT
SCHEMBL1575665 0.83 GRIN2B (0.56) GRIN2BTP53RAB9APOLBLMNA
SCHEMBL1575216 0.83 GRIN2B (0.58) GRIN2BTP53RAB9ALMNAMAPT
SCHEMBL1574971 0.83 ALDH1A1 (0.63) GRIN2BRAB9APOLBLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2308562-A2 Azetidine ring compounds and drugs comprising the same Ono Pharmaceutical Co., Ltd. (JP) 2011-04-13 EP disclosed
US-7511159-B2 Azetidine ring compounds and drugs comprising the same ONO PHARMACEUTICAL CO., LTD. (JP) 2009-03-31 US disclosed
US-20070135402-A1 Azetidine ring compounds and drugs comprising the same ONO PHARMACEUTICAL CO., LTD. (JP) 2007-06-14 US disclosed
EP-1698375-A1 AZETIDINE RING COMPOUNDS AND DRUGS COMPRISING THE SAME ONO PHARMACEUTICAL CO., LTD. (JP) 2006-09-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070135402-A1 Azetidine ring compounds and drugs comprising the same EDNRA, LIPG, EDNRB GRIN2B 3001/4885TP53 3220/4885RAB9A 898/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.