SCHEMBL1575615

SCHEMBL1575615

CC(C)CN(CC(C)C)C1CN(C(=O)NCc2ccccc2)C1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
KDM4E B2RXH2 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MEN1 O00255 3/20 0.49
NPSR1 Q6W5P4 2/20 0.49
ALDH1A1 P00352 3/20 0.47
HRH3 Q9Y5N1 2/20 0.47
MAPT P10636 1/20 0.46
RORC P51449 1/20 0.46
GAA P10253 1/20 0.45
GRIN2B Q13224 1/20 0.45
F2 P00734 1/20 0.44
PRSS1 P07477 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1574722 0.88 ALDH1A1 (0.47) KMT2AKDM4EL3MBTL1MEN1ALDH1A1
SCHEMBL1574418 0.85 KDM4E (0.57) KMT2AKDM4EMEN1NPSR1ALDH1A1
SCHEMBL1575097 0.84 KDM4E (0.52) KMT2AKDM4EL3MBTL1MEN1NPSR1
SCHEMBL1574975 0.83 KDM4E (0.54) KMT2AKDM4EMEN1NPSR1ALDH1A1
SCHEMBL1574791 0.82 KDM4E (0.56) KMT2AKDM4EMEN1NPSR1ALDH1A1
SCHEMBL1574846 0.82 NAMPT (0.50) KDM4EALDH1A1MAPTGRIN2B
SCHEMBL1575065 0.79 KDM4E (0.52) KMT2AKDM4EMEN1NPSR1ALDH1A1
SCHEMBL1575211 0.78 KMT2A (0.47) KMT2AMEN1ALDH1A1
SCHEMBL1574782 0.77 KDM4E (0.53) KMT2AKDM4EL3MBTL1MEN1NPSR1
SCHEMBL1575452 0.76 GAA (0.48) KMT2AKDM4EALDH1A1GAAGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2308562-A2 Azetidine ring compounds and drugs comprising the same Ono Pharmaceutical Co., Ltd. (JP) 2011-04-13 EP disclosed
US-7511159-B2 Azetidine ring compounds and drugs comprising the same ONO PHARMACEUTICAL CO., LTD. (JP) 2009-03-31 US disclosed
US-20070135402-A1 Azetidine ring compounds and drugs comprising the same ONO PHARMACEUTICAL CO., LTD. (JP) 2007-06-14 US disclosed
EP-1698375-A1 AZETIDINE RING COMPOUNDS AND DRUGS COMPRISING THE SAME ONO PHARMACEUTICAL CO., LTD. (JP) 2006-09-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070135402-A1 Azetidine ring compounds and drugs comprising the same EDNRA, LIPG, EDNRB KMT2A 2539/4885KDM4E 516/4885L3MBTL1 3473/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.