SCHEMBL15775100

SCHEMBL15775100

COc1cc(C(=O)O)cc2cc(Br)ccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA4 P22748 2/20 0.50
CA6 P23280 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
CA3 P07451 1/20 0.50
PKM P14618 1/20 0.50
CA5A P35218 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
TPMT P51580 2/20 0.49
PTGS2 P35354 1/20 0.47
POLB P06746 2/20 0.47
HTT P42858 1/20 0.46
RXFP1 Q9HBX9 3/20 0.44
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27619794 0.88 CA12 (0.50) CA12CA1CA2CA4CA6
SCHEMBL15774869 0.86 TSHR (0.53) POLBHTTRXFP1TUBB4ATUBB
SCHEMBL14217542 0.85 KDM4E (0.51) CA12CA1CA2CA4CA6
SCHEMBL15774677 0.81 HSD17B2 (0.52) CA12CA1CA2CA7CA9
SCHEMBL15775076 0.80 POLB (0.42) POLBRXFP1LMNASMN1; SMN2L3MBTL1
SCHEMBL18288064 0.79 ALOX15 (0.55) CA12CA1CA2CA4CA6
SCHEMBL10702559 0.76 HTT (0.56) CA12CA1CA2CA4CA6
SCHEMBL8960918 0.76 CA12 (0.62) CA12CA1CA2CA4CA6
SCHEMBL28857298 0.75 CA1 (0.69) CA12CA1CA2CA4CA6
SCHEMBL11507377 0.75 POLB (0.56) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014086697-A1 SUBSTITUTED THIAZOLE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2014-06-12 WO disclosed