SCHEMBL1583519

SCHEMBL1583519

Fc1ccc(-c2cncc(CNCCOc3cccc4cccnc34)c2)c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GLRA3 O75311 2/20 0.45
RAB9A P51151 2/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
KMT2A Q03164 1/20 0.43
KCNH2 Q12809 4/20 0.42
GRIN2B Q13224 3/20 0.42
NMT2 O60551 1/20 0.42
NMT1 P30419 1/20 0.42
GLRB P48167 1/20 0.40
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR1A P08908 2/20 0.39
MCHR1 Q99705 1/20 0.39
CYP2D6 P10635 1/20 0.39
ADRA1A P35348 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1582764 0.99 GLRA3 (0.45) GLRA3RAB9AMEN1NPC1KMT2A
SCHEMBL1583360 0.88 GLRA3 (0.47) GLRA3RAB9AMEN1NPC1KMT2A
SCHEMBL1583365 0.88 GLRA3 (0.51) GLRA3RAB9AMEN1NPC1KMT2A
SCHEMBL1582788 0.88 MEN1 (0.46) MEN1KMT2AKCNH2GRIN2BNMT2
Hydrochloric Acid SCHEMBL1582650 0.87 GLRA3 (0.46) GLRA3RAB9AMEN1NPC1KMT2A
Hydrochloric Acid SCHEMBL1582253 0.87 GLRA3 (0.50) GLRA3RAB9AMEN1NPC1KMT2A
Hydrochloric Acid SCHEMBL1582269 0.87 GLRA3 (0.50) GLRA3RAB9AMEN1NPC1KMT2A
Hydrochloric Acid SCHEMBL1582817 0.87 MEN1 (0.45) MEN1KMT2AKCNH2GRIN2BNMT2
SCHEMBL1583040 0.86 KCNH2 (0.43) KMT2AKCNH2GRIN2BNMT2NMT1
Hydrochloric Acid SCHEMBL1582866 0.86 ADRA1D (0.44) KMT2AKCNH2GRIN2BNMT2NMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1292592-B1 HETEROCYCLIC AMINOALKYL PYRIDINE DERIVATIVES AS PSYCHOPHARMACEUTICALS MERCK PATENT GMBH (DE) 2011-04-20 EP claimed
EP-1292592-B1 HETEROCYCLIC AMINOALKYL PYRIDINE DERIVATIVES AS PSYCHOPHARMACEUTICALS MERCK PATENT GMBH (DE) 2011-04-20 EP disclosed