SCHEMBL1584564

SCHEMBL1584564

O=C(c1nc2c(C(F)(F)F)cc(-c3ccoc3)cn2c1Cl)N1CCN(C2CCC2)C(=O)C1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 9/20 0.47
IRAK4 Q9NWZ3 1/20 0.35
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
ERN1 O75460 1/20 0.32
TYRO3 Q06418 1/20 0.32
MERTK Q12866 1/20 0.32
TRPV1 Q8NER1 1/20 0.31
KMT2A Q03164 1/20 0.31
RBP4 P02753 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1583038 0.98 P2RX7 (0.49) P2RX7IRAK4NPC1POLBRAB9A
SCHEMBL12720955 0.98 P2RX7 (0.48) P2RX7IRAK4NPC1POLBRAB9A
SCHEMBL12720597 0.98 P2RX7 (0.48) P2RX7IRAK4NPC1POLBRAB9A
SCHEMBL1583571 0.93 P2RX7 (0.41) P2RX7IRAK4TYRO3MERTKTRPV1
SCHEMBL1584096 0.92 P2RX7 (0.39) P2RX7ERN1TYRO3MERTKRBP4
SCHEMBL12720664 0.92 P2RX7 (0.40) P2RX7TYRO3MERTKTRPV1RBP4
SCHEMBL1583715 0.92 P2RX7 (0.38) P2RX7ERN1TYRO3MERTKTRPV1
SCHEMBL1583716 0.92 P2RX7 (0.38) P2RX7ERN1TYRO3MERTKTRPV1
SCHEMBL12720642 0.92 P2RX7 (0.39) P2RX7TYRO3MERTK
SCHEMBL1583748 0.91 P2RX7 (0.39) P2RX7TYRO3MERTKRBP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011041713-A2 PIPERAZINYL ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2011-04-07 WO claimed