SCHEMBL15865618

SCHEMBL15865618

CC(C)(C)OC(=O)c1cccc(CN(CCN(CC(=O)O)Cc2cccc(C(=O)OC(C)(C)C)n2)CC(=O)O)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
HPGDS O60760 1/20 0.35
PTGER2 P43116 4/20 0.34
BRD4 O60885 1/20 0.34
AKT1 P31749 1/20 0.33
MAPT P10636 1/20 0.33
SLC7A5 Q01650 1/20 0.33
MRGPRX4 Q96LA9 3/20 0.32
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32
SKP2 Q13309 1/20 0.32
PDE5A O76074 1/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15865612 0.90 CYP1A2 (0.36) CYP1A2HPGDSPTGER2BRD4AKT1
SCHEMBL2362585 0.88 MRGPRX4 (0.35) CYP1A2HPGDSPTGER2BRD4AKT1
SCHEMBL15865620 0.84 MRGPRX4 (0.33) CYP1A2BRD4AKT1MRGPRX4PDE5A
SCHEMBL23567539 0.84 NR1D1 (0.40) CYP1A2HPGDSBRD4AKT1MRGPRX4
SCHEMBL15865629 0.82 MRGPRX4 (0.39) CYP1A2MAPTMRGPRX4
SCHEMBL2349945 0.81 KDM4E (0.48) BRD4MRGPRX4
SCHEMBL29892650 0.81 KDM4E (0.48) BRD4MRGPRX4
SCHEMBL27119074 0.80 MRGPRX4 (0.37) CYP1A2HPGDSBRD4SLC7A5MRGPRX4
SCHEMBL30801055 0.80 MRGPRX4 (0.37) CYP1A2HPGDSBRD4SLC7A5MRGPRX4
SCHEMBL30960193 0.80 KDM4E (0.47) BRD4MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8772446-B2 Bifunctional chelating agents NORDION (CANADA) INC. (CA) 2014-07-08 US disclosed