SCHEMBL158662

SCHEMBL158662

NCC(=O)OC12CC3CC(CC(O)(C3)C1)C2

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
CYP19A1 P11511 2/20 0.37
ALDH1A1 P00352 3/20 0.37
HSD11B1 P28845 2/20 0.36
DPP4 P27487 4/20 0.36
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
EPHX2 P34913 1/20 0.34
CYP17A1 P05093 1/20 0.34
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28644764 1.00 PKM (0.42) PKMCYP19A1ALDH1A1HSD11B1DPP4
SCHEMBL4368869 0.83 PKM (0.38) PKMCYP19A1ALDH1A1HSD11B1DPP4
SCHEMBL5512258 0.83 PKM (0.38) PKMCYP19A1ALDH1A1HSD11B1DPP4
SCHEMBL2603060 0.83 HSD11B1 (0.41) PKMCYP19A1ALDH1A1HSD11B1DPP4
SCHEMBL158814 0.82 CYP19A1 (0.50) CYP19A1ALDH1A1EPHX2CYP17A1THRB
SCHEMBL14791585 0.81 PKM (0.46) PKMALDH1A1HSD11B1DPP4DPP8
SCHEMBL12936737 0.81 HSD11B1 (0.40) PKMCYP19A1ALDH1A1HSD11B1DPP4
Hydrochloric Acid SCHEMBL7313276 0.80 CYP19A1 (0.49) CYP19A1ALDH1A1EPHX2CYP17A1THRB
SCHEMBL18232632 0.80 MAPT (0.35) PKMCYP19A1ALDH1A1HSD11B1DPP4
SCHEMBL10228479 0.80 HSD11B1 (0.36) PKMCYP19A1ALDH1A1HSD11B1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611770-A1 PROCESS FOR THE REDUCTIVE AMINATION OF -KETO CARBOXYLIC ACIDS Sandoz AG (CH) 2013-07-10 EP disclosed
WO-2012028721-A1 PROCESS FOR THE REDUCTIVE AMINATION OF α-KETO CARBOXYLIC ACIDS SANDOZ AG (CH) 2012-03-08 WO disclosed