SCHEMBL15903276

SCHEMBL15903276

COc1cc2c(cc1OC)CC(C(=O)C1CCN(Cc3ccccc3)CC1)C2

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.65
DRD4 P21917 2/20 0.56
SIGMAR1 Q99720 2/20 0.56
ACHE P22303 2/20 0.56
FAAH O00519 1/20 0.56
ABCC4 O15439 1/20 0.56
CACNA1F O60840 1/20 0.56
PDE5A O76074 1/20 0.56
ABCB11 O95342 1/20 0.56
APP P05067 1/20 0.56
CHRM2 P08172 1/20 0.56
ABCB1 P08183 1/20 0.56
CYP3A4 P08684 1/20 0.56
CHRM5 P08912 1/20 0.56
ADRA2A P08913 1/20 0.56
CHRM1 P11229 1/20 0.56
ADRA2C P18825 1/20 0.56
SLC6A2 P23975 1/20 0.56
MAOB P27338 1/20 0.56
AGTR1 P30556 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3238921 0.99 BCHE (0.66) BCHEDRD4SIGMAR1ACHEFAAH
SCHEMBL27858398 0.84 BCHE (0.66) BCHEDRD4SIGMAR1ACHEFAAH
SCHEMBL27493904 0.83 ALDH1A1 (0.43) BCHEPDE4DDRD2KDM4ENPC1
SCHEMBL27608094 0.82 MEN1 (0.69) DRD4SIGMAR1ACHEFAAHDRD2
SCHEMBL29550512 0.79 BCHE (1.00) BCHEDRD4SIGMAR1ACHEFAAH
SCHEMBL13605247 0.79 BCHE (1.00) BCHEDRD4SIGMAR1ACHEFAAH
SCHEMBL28409804 0.78 BCHE (0.67) BCHEDRD4SIGMAR1ACHEFAAH
SCHEMBL16291177 0.78 MEN1 (0.68) SIGMAR1ACHEFAAHCHRM2
SCHEMBL2794872 0.75 ALDH1A1 (0.63) SIGMAR1KDM4E
SCHEMBL1475064 0.75 SIGMAR1 (0.71) DRD4SIGMAR1DRD2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2948429-A1 OXIDISABLE PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS ANTI-ALZHEIMER AGENTS INSA (Institut National des Sciences Appliquees) de Rouen (FR) 2015-12-02 EP disclosed
WO-2014114742-A1 OXIDISABLE PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS ANTI-ALZHEIMER AGENTS INSA (INSTITUT NATIONAL DES SCIENCES APPLIQUÉES) DE ROUEN (FR) 2014-07-31 WO disclosed