SCHEMBL15906147

SCHEMBL15906147

COc1cc(C)cc(Br)c1N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.55
NPSR1 Q6W5P4 1/20 0.55
L3MBTL1 Q9Y468 6/20 0.48
POLB P06746 2/20 0.48
ACHE P22303 2/20 0.48
ALDH1A1 P00352 1/20 0.42
CYP3A4 P08684 1/20 0.42
EP300 Q09472 1/20 0.40
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 3/20 0.38
GAA P10253 3/20 0.38
HPGD P15428 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ALOX5 P09917 1/20 0.36
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5028318 0.84 ACHE (0.59) MAPTNPSR1L3MBTL1POLBACHE
Hydrochloric Acid SCHEMBL8706033 0.81 ACHE (0.56) MAPTNPSR1L3MBTL1POLBACHE
SCHEMBL5946197 0.80 MAPT (0.57) MAPTNPSR1L3MBTL1POLBALDH1A1
SCHEMBL7479301 0.80 MAPT (0.57) MAPTNPSR1L3MBTL1POLBALDH1A1
SCHEMBL31211203 0.80 MAPT (0.57) MAPTNPSR1L3MBTL1POLBALDH1A1
SCHEMBL348577 0.78 MAPT (0.58) MAPTNPSR1ALDH1A1CYP3A4KDM4E
SCHEMBL1126364 0.77 ACHE (0.52) MAPTNPSR1L3MBTL1POLBACHE
SCHEMBL4730926 0.77 ALDH1A1 (0.56) MAPTNPSR1L3MBTL1POLBACHE
SCHEMBL30436671 0.77 ACHE (0.52) MAPTNPSR1L3MBTL1POLBACHE
SCHEMBL11139031 0.77 ACHE (0.52) MAPTNPSR1L3MBTL1POLBACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020015744-A1 AZAINDOLE DERIVATIVE AND USE THEREOF AS FGFR AND C-MET INHIBITOR 南京明德新药研发有限公司 2020-01-23 WO disclosed
US-8791267-B2 Biaryl PDE4 inhibitors for treating inflammatory, cardiovascular and CNS disorders DECODE GENETICS EHF (IS) 2014-07-29 US disclosed