SCHEMBL15919263

SCHEMBL15919263

CNC(=O)OCc1cc(-c2ccc(-c3ccc(-c4cc(C(C)=O)c5cnccc5n4)cc3)cc2)no1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.42
ESR2 Q92731 2/20 0.42
MAPT P10636 3/20 0.40
DHODH Q02127 3/20 0.37
CYP1A2 P05177 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 4/20 0.36
POLB P06746 2/20 0.36
LMNA P02545 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
PLA2G2A P14555 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15905447 0.91 GAA (0.45) MAPTDHODHSMN1; SMN2MEN1KMT2A
Hydrochloric Acid SCHEMBL15904893 0.90 GAA (0.44) MAPTDHODHSMN1; SMN2MEN1KMT2A
SCHEMBL17327503 0.90 MAPT (0.38) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL15919270 0.87 ACACB (0.42) MAPTSMN1; SMN2MEN1KMT2AKDM4E
SCHEMBL17323668 0.78 PLA2G2A (0.47) MAPTDHODHCYP1A2SMN1; SMN2MEN1
SCHEMBL15919268 0.78 SMN1; SMN2 (0.45) DHODHCYP1A2SMN1; SMN2MEN1KMT2A
SCHEMBL15919454 0.78 SMN1; SMN2 (0.57) MAPTDHODHCYP1A2SMN1; SMN2MEN1
SCHEMBL15919455 0.77 SMN1; SMN2 (0.56) DHODHCYP1A2SMN1; SMN2KMT2AALDH1A1
SCHEMBL15919272 0.77 PLA2G2A (0.46) MAPTDHODHCYP1A2SMN1; SMN2MEN1
SCHEMBL15905018 0.76 ALDH1A1 (0.43) MAPTCYP1A2SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014117090-A1 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2014-07-31 WO disclosed