SCHEMBL15925474

SCHEMBL15925474

Cc1sc(N2CCOCC2)nc1Cc1ccc2ccc(F)cc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.49
RAB9A P51151 4/20 0.49
NPC1 O15118 3/20 0.49
AR P10275 5/20 0.44
CYP3A4 P08684 5/20 0.43
PIK3CD O00329 4/20 0.43
PIK3CB P42338 4/20 0.43
PIK3CA P42336 1/20 0.43
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
KCNH2 Q12809 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
LMNA P02545 1/20 0.37
GRIA2 P42262 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15925464 0.97 SMN1; SMN2 (0.50) SMN1; SMN2RAB9ANPC1ARCYP3A4
SCHEMBL15925462 0.88 SMN1; SMN2 (0.49) SMN1; SMN2RAB9ANPC1ARCYP3A4
SCHEMBL15925455 0.87 AR (0.52) SMN1; SMN2RAB9ANPC1ARCYP3A4
SCHEMBL10288578 0.85 ALDH1A1 (0.47) SMN1; SMN2RAB9ANPC1ARCYP3A4
SCHEMBL15925487 0.85 CETP (0.48) SMN1; SMN2RAB9ANPC1ARPIK3CD
SCHEMBL15925488 0.84 AR (0.44) SMN1; SMN2RAB9ANPC1ARCYP3A4
SCHEMBL10298508 0.83 PIK3CD (0.61) SMN1; SMN2RAB9ANPC1CYP3A4PIK3CD
SCHEMBL15925471 0.83 SMN1; SMN2 (0.47) SMN1; SMN2RAB9ANPC1ARCYP3A4
SCHEMBL15925468 0.82 AR (0.44) SMN1; SMN2RAB9ANPC1ARCYP3A4
SCHEMBL15925466 0.82 CETP (0.49) SMN1; SMN2RAB9ANPC1ARPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796268-B2 Heteroaryls and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2014-08-05 US disclosed