SCHEMBL15925487

SCHEMBL15925487

COc1ccc2ccc(Cc3nc(N4CCOCC4)sc3C)cc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 1/20 0.48
APP P05067 1/20 0.46
AR P10275 1/20 0.42
PPARG P37231 2/20 0.42
PPARA Q07869 2/20 0.42
KDM4E B2RXH2 5/20 0.42
ALDH1A1 P00352 4/20 0.42
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPC1 O15118 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
RAB9A P51151 1/20 0.42
F2 P00734 1/20 0.41
F2RL3 Q96RI0 1/20 0.41
PIK3CD O00329 2/20 0.40
PIK3CA P42336 2/20 0.40
LMNA P02545 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15925466 0.98 CETP (0.49) CETPAPPARPPARGPPARA
SCHEMBL15925458 0.89 CETP (0.58) CETPAPPARPPARGPPARA
SCHEMBL15925455 0.88 AR (0.52) CETPARPPARGPPARAALDH1A1
SCHEMBL10288616 0.86 PIK3CD (0.48) CETPAPPKDM4EALDH1A1GAA
SCHEMBL15925474 0.85 SMN1; SMN2 (0.49) ARPPARGPPARAALDH1A1HPGD
SCHEMBL10298737 0.84 CETP (0.49) CETPAPPKDM4EALDH1A1HPGD
SCHEMBL15925464 0.84 SMN1; SMN2 (0.50) CETPARPPARGPPARAALDH1A1
SCHEMBL10288310 0.83 PIK3CD (0.50) CETPAPPKDM4EALDH1A1GAA
SCHEMBL15925468 0.83 AR (0.44) CETPARPPARGPPARAALDH1A1
SCHEMBL15925488 0.83 AR (0.44) CETPARPPARGPPARAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796268-B2 Heteroaryls and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2014-08-05 US disclosed