SCHEMBL15925699

SCHEMBL15925699

CC(=O)Nc1cc(-c2cc(C(O)c3ccc(Cl)cc3)c(-c3ncc[nH]3)s2)ccn1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.43
DBF4 Q9UBU7 1/20 0.43
PIK3C3 Q8NEB9 11/20 0.40
TGFBR1 P36897 1/20 0.37
TGFBR2 P37173 1/20 0.37
CNR1 P21554 1/20 0.37
CYP3A4 P08684 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
FFAR2 O15552 1/20 0.36
FPR2 P25090 1/20 0.35
NPC1 O15118 1/20 0.35
NR1I2 O75469 1/20 0.35
AHR P35869 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15925740 0.90 CDC7 (0.40) CDC7DBF4PIK3C3TGFBR1TGFBR2
SCHEMBL15925751 0.90 CDC7 (0.40) CDC7DBF4PIK3C3TGFBR1TGFBR2
SCHEMBL10288807 0.89 CDC7 (0.42) CDC7DBF4PIK3C3TGFBR1TGFBR2
SCHEMBL15925761 0.87 CDC7 (0.41) CDC7DBF4PIK3C3TGFBR1TGFBR2
SCHEMBL15925767 0.86 CDC7 (0.39) CDC7DBF4PIK3C3TGFBR1TGFBR2
SCHEMBL15925705 0.84 MAPK1 (0.35) FFAR2MAPK14
SCHEMBL15925723 0.84 MAPK1 (0.35) FFAR2MAPK14
SCHEMBL15925728 0.84 MAPK1 (0.35) FFAR2MAPK14
SCHEMBL15925694 0.84 IDO1 (0.32) FFAR2
SCHEMBL15925713 0.84 IDO1 (0.32) FFAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796271-B2 Heteroaryls and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2014-08-05 US disclosed