SCHEMBL15926258

SCHEMBL15926258

C=C/C=C\C=C(/C)NC(=O)CCC1c2c(F)cccc2C(=O)N1Cc1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
SIGMAR1 Q99720 5/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TSHR P16473 1/20 0.32
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2644689 0.77 MAPT (0.43) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL2643618 0.74 MAPT (0.40) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL27746396 0.74 ALDH1A1 (0.43) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL2643582 0.74 MAPT (0.40) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL2644105 0.74 MAPT (0.46) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL2643774 0.74 KDM4E (0.47) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL2643961 0.73 HTT (0.46) MAPTALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL2663945 0.73 MAPT (0.35) MAPTALDH1A1KDM4ESIGMAR1POLB
SCHEMBL2644848 0.73 MAPT (0.37) MAPTALDH1A1KDM4ESIGMAR1CYP1A2
SCHEMBL2644069 0.72 DRD4 (0.35) MAPTALDH1A1KDM4ESIGMAR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796313-B2 Substituted dihydroisoindolones as allosteric modulators of glucokinase JANSSEN PHARMACEUTICA N.V. (BE) 2014-08-05 US disclosed