SCHEMBL15943019

SCHEMBL15943019

Cc1ccc(-c2cc(C(=O)O)cc(-n3nnnc3C(C)F)c2)nc1

nearest known ligand 0.40

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 16/20 0.40
P2RX2 Q9UBL9 16/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10244810 0.85 P2RX3 (0.39) P2RX3P2RX2
SCHEMBL357241 0.82 NR1I2 (0.38) P2RX3P2RX2
SCHEMBL357773 0.80 ALDH1A1 (0.39) P2RX3P2RX2
SCHEMBL2269597 0.79 P2RX3 (0.42) P2RX3P2RX2
SCHEMBL4051058 0.77 P2RX3 (0.46) P2RX3P2RX2
SCHEMBL12200045 0.77 P2RX3 (0.40) P2RX3P2RX2
SCHEMBL4316321 0.77 P2RX3 (0.60) P2RX3P2RX2
SCHEMBL4323150 0.77 P2RX3 (0.59) P2RX3P2RX2
SCHEMBL4321379 0.77 NR1I2 (0.54) P2RX3P2RX2
SCHEMBL4565089 0.77 NR1I2 (0.36) P2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2570407-B1 TETRAZOLE-SUBSTITUTED ARYLAMIDE DERIVATIVES AND THEIR USE AS P2X3 AND/OR P2X2/3 PURINERGIC RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2014-08-13 EP disclosed