SCHEMBL15949103

SCHEMBL15949103

Cc1cc(F)ccc1[C@@H](C/C(=N\O)c1ccc(=O)[nH]c1C)c1ccc(-c2ccc(S(N)(=O)=O)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.35
CHRNA7 P36544 4/20 0.33
PTGS2 P35354 2/20 0.32
CA1 P00915 3/20 0.32
CA2 P00918 3/20 0.32
CA9 Q16790 3/20 0.32
CA12 O43570 2/20 0.32
CA14 Q9ULX7 1/20 0.32
BRD4 O60885 1/20 0.32
IKBKB O14920 1/20 0.32
CHUK O15111 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363176 0.81 GPBAR1 (0.39) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL364467 0.81 GPBAR1 (0.39) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL363016 0.81 GPBAR1 (0.39) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL15949059 0.80 GPBAR1 (0.37) GPBAR1
SCHEMBL1389857 0.79 GPBAR1 (0.40) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL1390246 0.79 GPBAR1 (0.40) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL1389860 0.79 GPBAR1 (0.40) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL1390245 0.79 GPBAR1 (0.40) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL1389930 0.79 GPBAR1 (0.40) GPBAR1CHRNA7CA1CA2CA9
SCHEMBL1389932 0.79 GPBAR1 (0.40) GPBAR1CHRNA7CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP disclosed