SCHEMBL15949059

SCHEMBL15949059

COC(=O)CNC(=O)c1ccc(-c2ccc(C(C/C(=N\O)c3ccc(=O)[nH]c3C)c3ccc(F)cc3C)cc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.37
SLC6A9 P48067 5/20 0.33
EPHX2 P34913 4/20 0.33
MAPK14 Q16539 1/20 0.33
SLC6A5 Q9Y345 2/20 0.33
MMP1 P03956 1/20 0.33
MAPK1 P28482 1/20 0.33
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
ULK1 O75385 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365164 0.91 GPBAR1 (0.37) GPBAR1MAPK1ADORA2AADORA2B
SCHEMBL363619 0.84 GPBAR1 (0.39) GPBAR1SLC6A9EPHX2MAPK14SLC6A5
SCHEMBL1390044 0.82 GPBAR1 (0.39) GPBAR1SLC6A9MAPK14SLC6A5MMP1
SCHEMBL1390040 0.82 GPBAR1 (0.39) GPBAR1SLC6A9MAPK14SLC6A5MMP1
SCHEMBL15949103 0.80 GPBAR1 (0.35) GPBAR1
SCHEMBL15949003 0.77 GPBAR1 (0.48) GPBAR1
SCHEMBL363976 0.76 GPBAR1 (0.41) GPBAR1SLC6A9EPHX2MAPK14SLC6A5
SCHEMBL15949284 0.75 GPBAR1 (0.60) GPBAR1
SCHEMBL1390253 0.75 GPBAR1 (0.41) GPBAR1SLC6A9SLC6A5MMP1
SCHEMBL1390250 0.75 GPBAR1 (0.41) GPBAR1SLC6A9SLC6A5MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP disclosed