SCHEMBL363176

SCHEMBL363176

Cc1cc(F)ccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(-c2ccc(S(N)(=O)=O)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.39
TDO2 P48775 1/20 0.35
CA1 P00915 10/20 0.34
CA2 P00918 10/20 0.34
CA9 Q16790 9/20 0.34
CA12 O43570 4/20 0.34
CA14 Q9ULX7 3/20 0.33
CA4 P22748 4/20 0.33
EPHX2 P34913 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
THRB P10828 1/20 0.32
CYP2C9 P11712 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363016 1.00 GPBAR1 (0.39) GPBAR1TDO2CA1CA2CA9
SCHEMBL364467 1.00 GPBAR1 (0.39) GPBAR1TDO2CA1CA2CA9
SCHEMBL363288 0.90 GPBAR1 (0.39) GPBAR1CA1CA2CA9CA12
SCHEMBL363235 0.88 GPBAR1 (0.51) GPBAR1EPHX2MEN1CYP1A2MAPK1
SCHEMBL365294 0.87 GPBAR1 (0.35) GPBAR1CA1CA2CA9CA12
SCHEMBL363976 0.82 GPBAR1 (0.41) GPBAR1EPHX2KDM4EMEN1ALDH1A1
SCHEMBL363293 0.82 GPBAR1 (0.39) GPBAR1MEN1ALDH1A1CYP1A2GAA
SCHEMBL1389930 0.82 GPBAR1 (0.40) GPBAR1CA1CA2CA9CA12
SCHEMBL1389857 0.82 GPBAR1 (0.40) GPBAR1CA1CA2CA9CA12
SCHEMBL1390246 0.82 GPBAR1 (0.40) GPBAR1CA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed