SCHEMBL15957129

SCHEMBL15957129

CN(C)CCS(=O)(=O)Nc1cc(O)cc(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 11/20 0.39
CA2 P00918 11/20 0.39
CA9 Q16790 11/20 0.39
CA12 O43570 1/20 0.39
CA3 P07451 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
THRA P10827 1/20 0.33
HIF1A Q16665 3/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488684 0.82 CA1 (0.42) CA1CA2CA9CA12CA3
SCHEMBL488838 0.81 CA1 (0.59) CA1CA2CA9CA12CA3
SCHEMBL15648519 0.79 CA1 (0.46) CA1CA2CA9CA12CA3
SCHEMBL15091821 0.73 CA1 (0.42) CA1CA2CA9CA12CA3
SCHEMBL488456 0.73 LIPG (0.41) CA1CA2CA9CA12CA3
SCHEMBL488760 0.72 CA1 (0.57) CA1CA2CA9CA12CA3
SCHEMBL21630366 0.72 CA1 (0.41) CA1CA2CA9CA12CA3
SCHEMBL21630389 0.72 CA1 (0.41) CA1CA2CA9CA12CA3
SCHEMBL8067182 0.72 CA1 (0.37) CA1CA2CA9CA12CA3
SCHEMBL15649508 0.71 CA1 (0.48) CA1CA2CA9CA12CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014124757-A1 PYRROLOTRIAZINE DERIVATIVES AS PI3K INHIBITORS ALMIRALL, S.A. (ES) 2014-08-21 WO disclosed