SCHEMBL15966747

SCHEMBL15966747

O=c1cc(-c2cccnc2)[nH]c2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 5/20 0.69
CTSL P07711 5/20 0.69
HPGD P15428 4/20 0.69
LMNA P02545 3/20 0.69
KDM4E B2RXH2 3/20 0.69
TUBB4A P04350 1/20 0.69
TP53 P04637 1/20 0.69
TUBB P07437 1/20 0.69
TUBA3C P0DPH7 1/20 0.69
TUBA1B P68363 1/20 0.69
TUBA4A P68366 1/20 0.69
TUBB4B P68371 1/20 0.69
TUBB3 Q13509 1/20 0.69
TUBB2A Q13885 1/20 0.69
TUBB8 Q3ZCM7 1/20 0.69
TUBA3E Q6PEY2 1/20 0.69
NPSR1 Q6W5P4 1/20 0.69
TUBA1A Q71U36 1/20 0.69
HSD17B10 Q99714 1/20 0.69
TUBA1C Q9BQE3 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6001723 0.83 CTSV (0.75) CTSVCTSLHPGDLMNAKDM4E
SCHEMBL367268 0.82 HPGD (1.00) CTSVCTSLHPGDLMNAKDM4E
SCHEMBL29411863 0.82 HPGD (1.00) CTSVCTSLHPGDLMNAKDM4E
SCHEMBL2789486 0.78 CYP19A1 (1.00) HPGDKDM4EHSD17B10CYP19A1RAB9A
SCHEMBL29790209 0.78 CYP19A1 (1.00) HPGDKDM4EHSD17B10CYP19A1RAB9A
Hydrochloric Acid SCHEMBL27830550 0.76 CYP19A1 (0.97) HPGDKDM4EHSD17B10CYP19A1RAB9A
SCHEMBL21563920 0.76 CYP19A1 (0.51) CYP19A1KMT2AADORA2AADORA1ALDH1A1
SCHEMBL26847017 0.76 CTSV (0.56) CTSVCTSLHPGDLMNAKDM4E
SCHEMBL2791999 0.76 CYP19A1 (0.59) LMNAKDM4ECYP19A1CYP11B1CYP11B2
Acetic Acid SCHEMBL6142950 0.75 HPGD (0.84) CTSVCTSLHPGDLMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014128206-A1 COMPOUNDS FOR USE IN INHIBITING HIV CAPSID ASSEMBLY Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-28 WO disclosed
WO-2014128206-A1 COMPOUNDS FOR USE IN INHIBITING HIV CAPSID ASSEMBLY Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-28 WO disclosed
EP-2769723-A1 Compounds for use in inhibiting HIV capsid assembly Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-27 EP disclosed
EP-2769723-A1 Compounds for use in inhibiting HIV capsid assembly Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-27 EP disclosed