SCHEMBL15967007

SCHEMBL15967007

Cn1cnc(OC(=O)N(CCc2cccc(C(F)(F)F)c2)CC2C3CNCC32)c1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 14/20 0.52
KCNH2 Q12809 8/20 0.44
SLC6A5 Q9Y345 4/20 0.41
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
CYP3A4 P08684 1/20 0.36
GPR52 Q9Y2T5 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15967281 0.92 SLC6A9 (0.59) SLC6A9KCNH2SLC6A5PSEN1PSEN2
Hydrochloric Acid SCHEMBL15967136 0.91 SLC6A9 (0.59) SLC6A9KCNH2SLC6A5PSEN1PSEN2
SCHEMBL15967219 0.87 SLC6A9 (0.63) SLC6A9KCNH2SLC6A5
SCHEMBL6105332 0.86 SLC6A9 (0.65) SLC6A9KCNH2SLC6A5CYP3A4CYP2D6
SCHEMBL15967152 0.85 SLC6A9 (0.52) SLC6A9KCNH2SLC6A5CYP3A4CYP2D6
SCHEMBL15967057 0.83 SLC6A9 (0.58) SLC6A9KCNH2SLC6A5CYP3A4CYP2D6
SCHEMBL15967139 0.83 SLC6A9 (0.49) SLC6A9KCNH2SLC6A5
SCHEMBL15967302 0.82 SLC6A9 (0.49) SLC6A9KCNH2SLC6A5
SCHEMBL15967170 0.82 SLC6A9 (0.52) SLC6A9KCNH2SLC6A5PSEN1PSEN2
SCHEMBL15966993 0.82 SLC6A9 (0.49) SLC6A9KCNH2SLC6A5CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869019-B1 BICYCLIC [3.1.0] HETEROARYL AMIDES AS TYPE I GLYCINE TRANSPORT INHIBITORS PFIZER PROD INC (US) 2014-08-27 EP claimed