SCHEMBL15975103

SCHEMBL15975103

CS(=O)(=O)NC(=O)c1cccc(Cc2c(-c3ccccc3)[nH]c3cc(C4CC4)ccc23)n1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.39
MCL1 Q07820 6/20 0.38
PDE2A O00408 1/20 0.38
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
TLR9 Q9NR96 6/20 0.36
TLR8 Q9NR97 5/20 0.36
TLR7 Q9NYK1 5/20 0.36
NR3C1 P04150 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11977719 0.92 BRD4 (0.38) BRD4PDE2AMTNR1AMTNR1BTLR9
SCHEMBL11979678 0.87 MCL1 (0.50) BRD4MCL1
SCHEMBL3708601 0.86 MTNR1A (0.39) PDE2AMTNR1AMTNR1BNR3C1
SCHEMBL11979686 0.86 MCL1 (0.50) BRD4MCL1
SCHEMBL4568428 0.86 TLR9 (0.41) PDE2AMTNR1AMTNR1BTLR9TLR8
SCHEMBL11978670 0.86 DGAT1 (0.41) PDE2AMTNR1AMTNR1BTLR9TLR7
SCHEMBL15975137 0.85 PDE2A (0.38) BRD4PDE2AMTNR1AMTNR1BTLR9
SCHEMBL15975092 0.84 MTNR1A (0.44) MCL1MTNR1AMTNR1B
SCHEMBL11978663 0.84 BRD4 (0.42) BRD4MCL1
SCHEMBL15975189 0.84 MCL1 (0.52) BRD4MCL1PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815903-B2 Indole derivative and pharmacologically acceptable salt thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2014-08-26 US disclosed
US-8815903-B2 Indole derivative and pharmacologically acceptable salt thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2014-08-26 US disclosed