SCHEMBL15975191

SCHEMBL15975191

CCS(=O)(=O)NC(=O)c1csc(Cc2c(-c3ccccc3)[nH]c3cc(OC)ccc23)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.49
MAPT P10636 6/20 0.48
LMNA P02545 5/20 0.48
ALDH1A1 P00352 3/20 0.48
RAB9A P51151 1/20 0.48
NPC1 O15118 1/20 0.48
CYP1A2 P05177 4/20 0.46
CYP3A4 P08684 4/20 0.46
CYP2C9 P11712 4/20 0.46
CYP2C19 P33261 4/20 0.46
POLB P06746 1/20 0.46
GAA P10253 1/20 0.43
ALOX12 P18054 1/20 0.43
MTNR1A P48039 3/20 0.42
MTNR1B P49286 3/20 0.42
CYP2D6 P10635 2/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 2/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4568231 0.86 SMN1; SMN2 (0.49) SMN1; SMN2MAPTLMNAALDH1A1RAB9A
SCHEMBL15975099 0.85 MTNR1A (0.43) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL3709879 0.84 MAPT (0.52) SMN1; SMN2MAPTLMNAALDH1A1RAB9A
SCHEMBL15975184 0.80 MTNR1A (0.41) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL15975186 0.80 MCL1 (0.35) SMN1; SMN2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL11977716 0.79 MTNR1A (0.44) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL11977720 0.79 TUBB4A (0.41) MAPTGAAKDM4ETUBB4ATUBB
SCHEMBL15975113 0.78 CYP19A1 (0.45) MAPTMTNR1AMTNR1BKDM4E
SCHEMBL15975135 0.78 MTNR1A (0.42) MAPTALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL15975092 0.78 MTNR1A (0.44) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815903-B2 Indole derivative and pharmacologically acceptable salt thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2014-08-26 US disclosed
US-8815903-B2 Indole derivative and pharmacologically acceptable salt thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2014-08-26 US disclosed