SCHEMBL15977013

SCHEMBL15977013

Fc1ccc(Nc2ccnc(-c3cccnc3)n2)cc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.52
MET P08581 1/20 0.52
CYP1A2 P05177 6/20 0.51
CLK4 Q9HAZ1 6/20 0.51
CYP3A4 P08684 5/20 0.51
CYP2C19 P33261 5/20 0.51
CYP2D6 P10635 4/20 0.51
ALOX15 P16050 3/20 0.51
KMT2A Q03164 3/20 0.50
DYRK1A Q13627 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
XBP1 P17861 1/20 0.50
STAT3 P40763 1/20 0.50
GSK3A P49840 1/20 0.50
GSK3B P49841 1/20 0.50
CDK5 Q00535 1/20 0.50
CDK5R1 Q15078 1/20 0.50
PPARG P37231 1/20 0.50
NR2E3 Q9Y5X4 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15966819 0.99 LMNA (0.51) LMNAMETCYP1A2CLK4CYP3A4
SCHEMBL15985696 0.88 LMNA (0.53) LMNACYP1A2CLK4CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL15966743 0.87 LMNA (0.52) LMNACYP1A2CLK4CYP3A4CYP2C19
SCHEMBL15977129 0.84 ABCG2 (0.57) LMNACYP1A2CLK4CYP3A4CYP2C19
SCHEMBL15985681 0.84 LMNA (0.53) LMNACYP1A2CLK4CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL15966688 0.83 LMNA (0.52) LMNACYP1A2CLK4CYP3A4CYP2C19
SCHEMBL15976914 0.82 CYP1A2 (0.43) LMNAMETCYP1A2CLK4CYP3A4
Hydrochloric Acid SCHEMBL15966824 0.81 CYP1A2 (0.43) LMNAMETCYP1A2CLK4CYP3A4
SCHEMBL15976947 0.79 LMNA (0.50) LMNACYP1A2CLK4CYP3A4CYP2C19
SCHEMBL15985701 0.79 LMNA (0.50) LMNACYP1A2CLK4CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014128213-A1 COMPOUNDS FOR USE IN INHIBITING HIV CAPSID ASSEMBLY Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-28 WO disclosed
EP-2769722-A1 Compounds for use in inhibiting HIV capsid assembly Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-27 EP disclosed