SCHEMBL15977129

SCHEMBL15977129

O=[N+]([O-])c1cc(Nc2ccnc(-c3cccnc3)n2)ccc1F

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 5/20 0.57
LMNA P02545 1/20 0.47
CYP1A2 P05177 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
XBP1 P17861 1/20 0.46
STAT3 P40763 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
CDK5 Q00535 1/20 0.46
CDK5R1 Q15078 1/20 0.46
KMT2A Q03164 2/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
ABL1 P00519 1/20 0.46
EGFR P00533 1/20 0.46
BCR P11274 1/20 0.46
SRC P12931 1/20 0.46
PRKCA P17252 1/20 0.46
PPARG P37231 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15977013 0.84 LMNA (0.52) LMNACYP1A2SMN1; SMN2XBP1STAT3
Hydrochloric Acid SCHEMBL15966819 0.83 LMNA (0.51) LMNACYP1A2SMN1; SMN2XBP1STAT3
SCHEMBL3858988 0.83 ABL1 (0.67) ABL1EGFRBCRSRCPRKCA
SCHEMBL655435 0.81 NPC1 (0.55) ABCG2LMNAGSK3AGSK3BCDK5
SCHEMBL15985696 0.78 LMNA (0.53) LMNACYP1A2SMN1; SMN2XBP1STAT3
Hydrochloric Acid SCHEMBL15966743 0.77 LMNA (0.52) LMNACYP1A2SMN1; SMN2XBP1STAT3
SCHEMBL15985701 0.74 LMNA (0.50) LMNACYP1A2SMN1; SMN2XBP1STAT3
SCHEMBL1980117 0.74 CYP11B1 (0.51) LMNACYP1A2MAPTHTTCYP3A4
Hydrochloric Acid SCHEMBL15966787 0.73 LMNA (0.49) LMNACYP1A2SMN1; SMN2XBP1STAT3
SCHEMBL15966858 0.72 AURKA (0.63) LMNACYP1A2SMN1; SMN2XBP1STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014128206-A1 COMPOUNDS FOR USE IN INHIBITING HIV CAPSID ASSEMBLY Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-28 WO disclosed
EP-2769723-A1 Compounds for use in inhibiting HIV capsid assembly Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-27 EP disclosed