SCHEMBL15977201

SCHEMBL15977201

Cc1ccc2c3c([nH]c2c1)CCN(C)C3

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.76
CHRNA7 P36544 1/20 0.66
SIRT2 Q8IXJ6 1/20 0.62
ALOX15 P16050 2/20 0.56
HSD17B10 Q99714 2/20 0.56
USP2 O75604 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
ACHE P22303 4/20 0.54
GRIN1 Q05586 3/20 0.54
GRIN2A Q12879 3/20 0.54
GRIN2D O15399 2/20 0.54
GRIN3B O60391 2/20 0.54
GRIN2B Q13224 2/20 0.54
GRIN2C Q14957 2/20 0.54
GRIN3A Q8TCU5 2/20 0.54
BAZ2B Q9UIF8 1/20 0.51
HTR6 P50406 2/20 0.51
KDM4E B2RXH2 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25512689 0.89 L3MBTL1 (0.61) L3MBTL1CHRNA7SIRT2CYP1A2CYP2D6
Dehydrostobadine SCHEMBL167500 0.88 L3MBTL1 (0.97) L3MBTL1CHRNA7SIRT2ALOX15HSD17B10
Dehydrostobadine SCHEMBL29468212 0.88 L3MBTL1 (0.97) L3MBTL1CHRNA7SIRT2ALOX15HSD17B10
SCHEMBL18034956 0.88 KDM4E (0.66) L3MBTL1CHRNA7SIRT2ALOX15HSD17B10
Dehydrostobadine SCHEMBL2837548 0.87 L3MBTL1 (1.00) L3MBTL1CHRNA7SIRT2ALOX15HSD17B10
Dehydrostobadine SCHEMBL3715610 0.87 L3MBTL1 (1.00) L3MBTL1CHRNA7SIRT2ALOX15HSD17B10
SCHEMBL2185371 0.84 CHRNA7 (0.64) L3MBTL1CHRNA7SIRT2ALOX15HSD17B10
SCHEMBL27099161 0.84 CHRNA7 (0.64) L3MBTL1CHRNA7SIRT2ALOX15HSD17B10
SCHEMBL168351 0.84 CHRNA7 (0.64) L3MBTL1CHRNA7SIRT2ALOX15HSD17B10
SCHEMBL167846 0.82 CHRNA7 (0.62) L3MBTL1CHRNA7SIRT2ALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019074979-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF GIRAFPHARMA, LLC (US) 2019-04-18 WO disclosed
EP-2476680-B1 (1-Azinone)-Substituted Pyridoindoles ALBANY MOLECULAR RES INC (US) 2014-08-27 EP disclosed