SCHEMBL15979679

SCHEMBL15979679

Cc1cc(C(=O)CCC(=O)c2cc(Cl)sc2Cl)c(Cl)s1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.61
DAO P14920 1/20 0.52
MAPT P10636 2/20 0.47
HPGD P15428 2/20 0.47
KDM4E B2RXH2 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
RAB9A P51151 3/20 0.41
NPC1 O15118 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
KDR P35968 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15988630 0.89 GSK3B (0.74) GSK3BDAOMAPTHPGDKDM4E
SCHEMBL19341288 0.86 GSK3B (0.61) GSK3BDAOMAPTHPGDKDM4E
SCHEMBL6802262 0.82 GSK3B (0.65) GSK3BDAOMAPTHPGDKDM4E
SCHEMBL10512352 0.78 GSK3B (0.69) GSK3BDAOMAPTHPGDKDM4E
SCHEMBL11847449 0.76 DAO (0.52) GSK3BDAOMAPTHPGDKDM4E
SCHEMBL6790563 0.76 GSK3B (1.00) GSK3BDAOMAPTHPGDKDM4E
SCHEMBL5725649 0.74 GSK3B (0.69) GSK3BDAOMAPTHPGDKDM4E
SCHEMBL8629968 0.74 DAO (0.63) GSK3BDAOMAPTHPGDKDM4E
SCHEMBL17929703 0.73 GSK3B (0.53) GSK3BDAOMAPTHPGDKDM4E
SCHEMBL13602654 0.73 GSK3B (0.49) GSK3BDAOMAPTHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11673885-B2 γ-diketones as Wnt/β-catenin signaling pathway activators BIOSPLICE THERAPEUTICS, INC. (US) 2023-06-13 US disclosed
US-9951053-B2 γ-diketones as Wnt/β-catenin signaling pathway activators SAMUMED, LLC (US) 2018-04-24 US disclosed
US-20170260176-A1 GAMMA-DIKETONES AS WNT/BETA -CATENIN SIGNALING PATHWAY ACTIVATORS MED-PATHWAYS II LIMITED (VG) 2017-09-14 US disclosed
US-9533976-B2 γ-diketones as WNT/β-catenin signaling pathway activators SAMUMED, LLC (US) 2017-01-03 US disclosed
US-20140243349-A1 GAMMA-DIKETONES AS WNT/BETA -CATENIN SIGNALING PATHWAY ACTIVATORS VICKERS VENTURE FUND VI PTE. LTD. (SG) 2014-08-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170260176-A1 GAMMA-DIKETONES AS WNT/BETA -CATENIN SIGNALING PATHWAY ACTIVATORS GSK3A, GSK3B, WNT1 GSK3B 2/4885DAO 3651/4885MAPT 395/4885
US-20140243349-A1 GAMMA-DIKETONES AS WNT/BETA -CATENIN SIGNALING PATHWAY ACTIVATORS GSK3A, GSK3B, WNT1 GSK3B 2/4885DAO 3651/4885MAPT 395/4885
US-11673885-B2 γ-diketones as Wnt/β-catenin signaling pathway activators GSK3A, GSK3B, WNT1 GSK3B 2/4885DAO 3757/4885MAPT 388/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.