Epiryanodine

Epiryanodine

SCHEMBL159872

CC(C)[C@@]1(O)[C@@H](OC(=O)c2ccc[nH]2)[C@@]2(O)[C@@]3(C)C[C@]4(O)O[C@@]5([C@H](O)[C@@H](C)CC[C@]35O)[C@@]2(O)[C@@]14C.CC(C)[C@@]1(O)[C@@H](OC(=O)c2ccc[nH]2)[C@@]2(O)[C@@]3(C)C[C@]4(O)O[C@@]5([C@H](O)[C@@H](C)CC[C@]35O)[C@@]2(O)[C@@]14C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
RYR1 P21817 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Epiryanodine SCHEMBL5933502 1.00 RYR1 (1.00) RYR1
Epiryanodine SCHEMBL20100627 1.00 RYR1 (1.00) RYR1
Epiryanodine SCHEMBL118946 1.00 RYR1 (1.00) RYR1
Epiryanodine SCHEMBL13912554 1.00 RYR1 (1.00) RYR1
Epiryanodine SCHEMBL20104624 1.00 RYR1 (1.00) RYR1
Epiryanodine SCHEMBL31236365 1.00 RYR1 (1.00) RYR1
Epiryanodine SCHEMBL25722480 1.00 RYR1 (1.00) RYR1
Epiryanodine SCHEMBL13479886 1.00 RYR1 (1.00) RYR1
Epiryanodine SCHEMBL5820916 0.99 RYR1 (0.98) RYR1
Epiryanodine SCHEMBL4318989 0.99 RYR1 (0.98) RYR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4117432-A2 FUNGICIDAL HALOMETHYL KETONES AND HYDRATES AND THEIR MIXTURES FMC CORPORATION (US) 2023-01-18 EP disclosed
WO-2021183707-A2 FUNGICIDAL HALOMETHYL KETONES AND HYDRATES AND THEIR MIXTURES FMC CORPORATION (US) 2021-09-16 WO disclosed
EP-3644731-A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO Dow AgroSciences LLC (US) 2020-05-06 EP disclosed
WO-2019005517-A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO DOW AGROSCIENCES LLC (US) 2019-01-03 WO disclosed
WO-2017062729-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2017-04-13 WO disclosed
WO-2016144351-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2016-09-15 WO disclosed
EP-3044220-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES E. I. du Pont de Nemours and Company (US) 2016-07-20 EP disclosed
EP-2999695-A1 SOLID FORMS OF FUNGICIDAL PYRAZOLES E. I. du Pont de Nemours and Company (US) 2016-03-30 EP disclosed
EP-2864327-A1 SOLID FORMS OF A PYRIDO-PYRIMIDINIUM INNER SALT E. I. Du Pont de Nemours and Company (US) 2015-04-29 EP disclosed
EP-2850074-A1 1,3-DIARYL-SUBSTITUTED HETEROCYCLIC PESTICIDES E. I. Du Pont de Nemours and Company (US) 2015-03-25 EP disclosed
WO-2013055584-A1 SOLID FORMS OF NEMATOCIDAL SULFONAMIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2013-04-18 WO disclosed
EP-2576523-A1 CRYSTALLINE FORM OF 4- [5 - [3 -CHLORO-5 - (TRIFLUOROMETHYL) PHENYL]-4, 5 - DIHYDRO - 5 - (TRIFLUOROMETHYL) -3 - ISOXAZOLYL]-N- [2-0X0-2- [ ( 2, 2, 2 - TRIFLUOROETHYL) AMINO]ETHYL]-1- NAPHTHALENECARBOXAMIDE E.I. DU PONT DE NEMOURS AND COMPANY (US) 2013-04-10 EP disclosed
WO-2012106495-A1 MESOIONIC PESTICIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-08-09 WO disclosed
WO-2012092115-A1 MESOIONIC PYRIDO [1,2 -A] PYRIMIDINE PESTICIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-07-05 WO disclosed
WO-2012087630-A1 PYRIDINE AND PYRIMIDINE COMPOUNDS FOR CONTROLLING INVERTEBRATE E.I. DU PONT DE NEMOURS AND COMPANY (US) 2012-06-28 WO disclosed
WO-2012054233-A1 NEMATOCIDAL SULFONAMIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-04-26 WO disclosed
WO-2012031061-A2 FUNGICIDAL PYRAZOLES AND THEIR MIXTURES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-03-08 WO disclosed
WO-2012012366-A1 PESTICIDAL 3-(ARYLOXY)AZACYCLOALKANES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-01-26 WO disclosed
WO-2011149749-A1 CRYSTALLINE FORM OF 4- [5 - [3 -CHLORO-5 - (TRIFLUOROMETHYL) PHENYL] -4, 5 - DIHYDRO - 5 - (TRIFLUOROMETHYL) -3 - ISOXAZOLYL] -N- [2-0X0-2- [ ( 2, 2, 2 - TRIFLUOROETHYL) AMINO] ETHYL] -1- NAPHTHALENECARBOXAMIDE E.I. DU PONT DE NEMOURS AND COMPANY (US) 2011-12-01 WO disclosed
WO-2011056463-A2 FUNGICIDAL MIXTURES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-05-12 WO disclosed