SCHEMBL16004304

SCHEMBL16004304

CN(C)CCOCc1ccc2c(c1)CN(C(=O)Cc1ccc(Cl)cc1)CCO2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.43
GPR142 Q7Z601 1/20 0.40
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ME2 P23368 1/20 0.37
ME1 P48163 1/20 0.37
ME3 Q16798 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
KMT2A Q03164 2/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
USP9X Q93008 1/20 0.36
GFER P55789 1/20 0.35
ATM Q13315 1/20 0.35
RAB9A P51151 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004305 0.91 RIPK1 (0.46) RIPK1GPR142L3MBTL1ME2ME1
SCHEMBL16003975 0.90 ABCB1 (0.46) RIPK1GPR142KMT2AGFERRAB9A
SCHEMBL16004306 0.89 RIPK1 (0.43) RIPK1GPR142ME2ME1ME3
SCHEMBL16003979 0.85 RIPK1 (0.41) RIPK1GPR142TSHRME2ME1
SCHEMBL16004134 0.84 ABCB1 (0.48) RIPK1GPR142KMT2AALDH1A1ABCB1
SCHEMBL16003981 0.80 PIK3CA (0.44) RIPK1GPR142KMT2A
SCHEMBL16003977 0.79 MEN1 (0.48) RIPK1GPR142KMT2A
SCHEMBL16004308 0.79 ABCB1 (0.48) RIPK1GPR142L3MBTL1KMT2AGFER
SCHEMBL16003983 0.78 GAA (0.43) RIPK1KMT2ACYP2C9CYP2C19RAB9A
SCHEMBL16004248 0.77 ABCB1 (0.50) RIPK1GPR142L3MBTL1KMT2AGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed