SCHEMBL16004134

SCHEMBL16004134

COc1ccc(CC(=O)N2CCOc3ccc(COCc4ccc(Cl)cc4)cc3C2)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.48
ABCC1 P33527 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
MAPT P10636 3/20 0.47
RIPK1 Q13546 2/20 0.43
THRB P10828 2/20 0.43
TP53 P04637 1/20 0.43
HPGD P15428 3/20 0.42
GAA P10253 1/20 0.42
CREBBP Q92793 1/20 0.41
RYR2 Q92736 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GPR142 Q7Z601 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16003977 0.91 MEN1 (0.48) MAPTRIPK1KMT2AGPR142
SCHEMBL16004248 0.89 ABCB1 (0.50) ABCB1ABCC1SMN1; SMN2MAPTRIPK1
SCHEMBL16004253 0.89 SMN1; SMN2 (0.54) ABCB1ABCC1SMN1; SMN2MAPTRIPK1
SCHEMBL16004247 0.89 HPGD (0.51) SMN1; SMN2MAPTRIPK1THRBTP53
SCHEMBL16004308 0.88 ABCB1 (0.48) ABCB1ABCC1SMN1; SMN2MAPTRIPK1
SCHEMBL16004136 0.86 GPR142 (0.46) ABCB1ABCC1SMN1; SMN2MAPTRIPK1
SCHEMBL16004238 0.86 ABCB1 (0.47) ABCB1ABCC1SMN1; SMN2MAPTRIPK1
SCHEMBL16004306 0.85 RIPK1 (0.43) MAPTRIPK1GAAALDH1A1KMT2A
SCHEMBL16003975 0.85 ABCB1 (0.46) ABCB1ABCC1SMN1; SMN2MAPTRIPK1
SCHEMBL16004091 0.84 ALDH1A1 (0.48) ABCB1ABCC1SMN1; SMN2MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed