SCHEMBL16022086

SCHEMBL16022086

CN(c1ccc2ncccc2c1)c1nc(Cl)ncc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DOT1L Q8TEK3 1/20 0.51
PIN1 Q13526 12/20 0.42
MAPT P10636 3/20 0.40
PDE10A Q9Y233 1/20 0.37
ALDH1A1 P00352 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NCOA1 Q15788 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
GFER P55789 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37
TUBB2A Q13885 1/20 0.37
TUBB8 Q3ZCM7 1/20 0.37
TUBA3E Q6PEY2 1/20 0.37
TUBA1A Q71U36 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1917609 0.77 PIN1 (0.52) PIN1MAPTL3MBTL1
SCHEMBL16012092 0.74 PIN1 (0.64) PIN1MAPTALDH1A1
SCHEMBL8297040 0.73 PIN1 (0.47) PIN1MAPTALDH1A1
SCHEMBL30366419 0.72 PIN1 (0.43) PIN1MAPTTUBB4ATUBBTUBA3C
SCHEMBL3394316 0.71 PIN1 (0.48) PIN1
SCHEMBL16513289 0.69 ABCG2 (0.52) PIN1MAPTALDH1A1
SCHEMBL30635859 0.69 ABCG2 (0.52) PIN1MAPTALDH1A1
SCHEMBL28787349 0.69 PIN1 (0.46) PIN1MAPT
SCHEMBL10810225 0.69 MEN1 (0.51) MAPTPDE10AALDH1A1L3MBTL1NCOA1
SCHEMBL13166210 0.68 ABCG2 (0.51) PIN1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014135244-A1 TRIAZOLO[4,5-D]PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF DISEASES SUCH AS CANCER MERCK PATENT GMBH (DE) 2014-09-12 WO disclosed