Guaifenesin

Guaifenesin

SCHEMBL160234

COc1ccccc1OC[C@@H](O)CO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 1.00
LMNA P02545 3/20 1.00
AGTR1 P30556 1/20 1.00
KDM4E B2RXH2 4/20 0.69
SMN1; SMN2 Q16637 3/20 0.64
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
CYP2C19 P33261 1/20 0.60
TSHR P16473 3/20 0.56
MAPK1 P28482 1/20 0.56
IDO1 P14902 1/20 0.54
ALDH1A1 P00352 1/20 0.54
HPGD P15428 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
MAPT P10636 1/20 0.51
CASR P41180 1/20 0.50
ALOX15 P16050 1/20 0.50
THRB P10828 1/20 0.49
HTT P42858 1/20 0.49
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Guaifenesin SCHEMBL29759010 1.00 CYP1A2 (1.00) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2
Guaifenesin SCHEMBL31161209 1.00 CYP1A2 (1.00) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2
Guaifenesin SCHEMBL4322 1.00 CYP1A2 (1.00) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2
Guaifenesin SCHEMBL4321 1.00 CYP1A2 (1.00) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2
Guaifenesin SCHEMBL4894727 0.98 CYP1A2 (0.96) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2
Guaifenesin SCHEMBL2459821 0.98 CYP1A2 (0.96) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2
Guaifenesin SCHEMBL28898302 0.92 CYP1A2 (0.84) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2
Guaifenesin SCHEMBL28062894 0.92 CYP1A2 (0.84) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2
SCHEMBL29941729 0.90 LMNA (0.82) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2
SCHEMBL2328960 0.90 LMNA (0.82) CYP1A2LMNAAGTR1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1765 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026104828-A1 INCONTINENCE MANAGEMENT DEVICE JOYVIÉ HEALTH LTD (GB) 2026-05-21 WO claimed
EP-4687591-A1 RESILIENT UNIT AND METHOD OF MANUFACTURE HS Products Limited (GB) 2026-02-11 EP claimed
WO-2025264590-A1 METHOD FOR IMPROVED SENSITIVITY OF INTEGRITY TESTS OF FILTERS IN ASSEMBLIES EMD MILLIPORE CORPORATION (US) 2025-12-26 WO claimed
EP-4655036-A1 CATHETER KIT CLINISUPPLIES LIMITED (GB) 2025-12-03 EP claimed
EP-4649214-A1 MANUAL CONCRETE FINISHING TOOLS AND COMPONENTS FOR USE THEREWITH Baron Innovative Technology LP (US) 2025-11-19 EP claimed
EP-4637434-A1 CAP ASSEMBLY FOR AEROSOL GENERATING DEVICE Imperial Tobacco Limited (GB) 2025-10-29 EP claimed
WO-2025202225-A1 SYRINGE SURROGATE AND METHOD OF TESTING AN AUTOINJECTOR F. HOFFMANN-LA ROCHE AG (CH) 2025-10-02 WO claimed
CN-119962831-A Mangrove ecological system health evaluation method and system based on species level 广东省林业科学研究院 2025-05-09 CN claimed
WO-2025093847-A1 EAR INSERT FLARE AUDIO TECHNOLOGIES LIMITED (GB) 2025-05-08 WO claimed
EP-4543506-A1 AN EXTENDED DURATION INFUSION SYSTEM University of Galway (IE) 2025-04-30 EP claimed
EP-0032926-A4 ELECTRIC-HYDRAULIC DRIVE MODULES FOR VEHICLES. PACCAR INC (US) 1981-12-16 EP claimed
WO-1981002861-A1 WORKPIECE CLAMP MERCER NAIRNE & CO LTD (GB) 1981-10-15 WO claimed
EP-0035497-A1 SEAL ASSEMBLY. CATERPILLAR TRACTOR CO (US) 1981-09-16 EP claimed
EP-0032926-A1 ELECTRIC-HYDRAULIC DRIVE MODULES FOR VEHICLES. PACCAR INC (US) 1981-08-05 EP claimed
EP-0030536-A1 INK DELIVERY APPARATUS FOR A DOT MATRIX PRINTER CENTRONICS DATA COMPUTER CORPORATION (US) 1981-06-24 EP claimed
WO-1981001211-A1 SECURITY VALIDATOR ARDAC INC (US) 1981-04-30 WO claimed
WO-1981000699-A1 SEAL ASSEMBLY CATERPILLAR TRACTOR CO (US) 1981-03-19 WO claimed
WO-1981000382-A1 ELECTRIC-HYDROSTATIC DRIVE MODULES FOR VEHICLES PACCAR INC (US) 1981-02-19 WO claimed
WO-1980002673-A1 INK DELIVERY APPARATUS FOR A DOT MATRIX PRINTER CENTRONICS DATA COMPUTER (US) 1980-12-11 WO claimed
WO-1980002676-A1 WINDOW CLIP RETAINER GARMAN R 1980-12-11 WO claimed