SCHEMBL16023965

SCHEMBL16023965

COc1ccc(CN(C)c2nc(N=O)nn2Cc2ccc(OC)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
APLNR P35414 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
HTT P42858 1/20 0.39
CMA1 P23946 1/20 0.38
NPBWR1 P48145 3/20 0.38
ADORA2A P29274 2/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
KDM4E B2RXH2 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
CACNA1G O43497 1/20 0.36
CACNA1H O95180 1/20 0.36
CACNA1I Q9P0X4 1/20 0.36
MCHR1 Q99705 1/20 0.36
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16014680 0.81 ALDH1A1 (0.52) ALDH1A1APLNRSMN1; SMN2HTTCMA1
SCHEMBL16014406 0.79 MAPT (0.46) ALDH1A1APLNRSMN1; SMN2HTTCMA1
SCHEMBL17403441 0.77 ACP1 (0.44) ALDH1A1SMN1; SMN2ADORA2AMEN1KMT2A
SCHEMBL16023894 0.75 SMN1; SMN2 (0.38) ALDH1A1SMN1; SMN2NPBWR1ADORA2AMAPT
SCHEMBL18723727 0.70 PIK3CA (0.43) ALDH1A1APLNRSMN1; SMN2HTTCMA1
SCHEMBL15556570 0.69 ALDH1A1 (0.44) ALDH1A1APLNRCMA1NPBWR1ADORA2A
SCHEMBL15556088 0.69 MAPT (0.40) ALDH1A1APLNRSMN1; SMN2HTTCMA1
SCHEMBL15606508 0.68 PIK3CA (0.43) ALDH1A1APLNRSMN1; SMN2HTTCMA1
SCHEMBL15556714 0.68 MAPT (0.47) APLNRSMN1; SMN2CMA1NPBWR1MAPT
SCHEMBL16014845 0.66 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2HTTCMA1NPBWR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014135472-A1 ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2014-09-12 WO disclosed