SCHEMBL16063576

SCHEMBL16063576

CCNNC(=O)[C@@H](Cc1ccc(O)cc1)NC(C)=O

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.54
CTSS P25774 1/20 0.48
CTSK P43235 1/20 0.48
CPA1 P15085 2/20 0.47
MME P08473 1/20 0.47
ACE P12821 1/20 0.47
ACE2 Q9BYF1 1/20 0.47
CPA2 P48052 1/20 0.46
CPA4 Q9UI42 1/20 0.46
CTSL P07711 1/20 0.45
FOLH1 Q04609 1/20 0.45
OPRD1 P41143 2/20 0.45
OPRM1 P35372 1/20 0.45
OPRK1 P41145 1/20 0.45
CHRND Q07001 5/20 0.44
CHRNA1 P02708 1/20 0.44
CHRNG P07510 1/20 0.44
CHRNB1 P11230 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5009890 0.87 GRIA1 (0.62) GRIA1CTSSCTSKCPA1MME
SCHEMBL5007773 0.87 GRIA1 (0.62) GRIA1CTSSCTSKCPA1MME
SCHEMBL16116805 0.86 ACACB (0.51)
SCHEMBL18647567 0.85 ACACB (0.55)
SCHEMBL16116808 0.85 GRIA1 (0.56) GRIA1CTSSCTSKCPA1MME
SCHEMBL30493613 0.84 GRIA1 (0.55) GRIA1CTSSCTSKCPA1MME
SCHEMBL25139820 0.83 GRIA1 (0.57) GRIA1CTSSCTSKCPA1MME
SCHEMBL24724924 0.83 GRIA1 (0.57) GRIA1CTSSCTSKCPA1MME
SCHEMBL12632559 0.83 GRIA1 (0.57) GRIA1CTSSCTSKCPA1MME
SCHEMBL6862498 0.83 GRIA1 (0.57) GRIA1CTSSCTSKCPA1MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015077303-A1 PATIENT SELECTION METHOD FOR INFLAMMATION PURDUE RESEARCH FOUNDATION (US) 2015-05-28 WO disclosed
WO-2014149073-A1 METHODS OF MANUFACTURE AND SYNTHESIS OF AMINO ACID LINKING GROUPS CONJUGATED TO COMPOUNDS USED FOR TARGETED IMAGING OF TUMORS ON TARGET LABORATORIES LLC (US) 2014-09-25 WO disclosed
WO-2014149069-A1 SYNTHESIS AND COMPOSITION OF AMINO ACID LINKING GROUPS CONJUGATED TO COMPOUNDS USED FOR THE TARGETED IMAGING OF TUMORS PURDUE RESEARCH FOUNDATION (US) 2014-09-25 WO disclosed
WO-2014143309-A1 FLUORESCENCE IMAGING OF INFLAMMATORY DISEASES PURDUE RESEARCH FOUNDATION (US) 2014-09-18 WO disclosed